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- [31] Androgen receptor degradation by the proteolysis-targeting chimera ARCC-4 outperforms enzalutamide in cellular models of prostate cancer drug resistanceCommunications Biology, 1Jemilat Salami论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyShanique Alabi论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyRyan R. Willard论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyNick J. Vitale论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyJing Wang论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyHanqing Dong论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyMeizhong Jin论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyDonald P. McDonnell论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyAndrew P. Crew论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyTaavi K. Neklesa论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental BiologyCraig M. Crews论文数: 0 引用数: 0 h-index: 0机构: Yale University,Department of Molecular, Cellular and Developmental Biology
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- [33] Discovery of Selective Proteolysis-Targeting Chimera Degraders Targeting PTP1B as Long-Term Hypoglycemic AgentsJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (09) : 7569 - 7584Yang, Zunhua论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaYing, Yuqi论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaCheng, Shaobing论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Natl Engn Res Ctr Mfg Technol TCM Solid Preparat, Nanchang 330006, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaWu, Jiamin论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Natl Engn Res Ctr Mfg Technol TCM Solid Preparat, Nanchang 330006, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaZhang, Ziwei论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaHu, Pei论文数: 0 引用数: 0 h-index: 0机构: Jiangzhong Pharmaceut Co Ltd, Nanchang 330103, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaXiong, Jian论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaLi, Huilan论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Natl Engn Res Ctr Mfg Technol TCM Solid Preparat, Nanchang 330006, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaZeng, Qing论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaCai, Zhifang论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaFeng, Yulin论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Natl Engn Res Ctr Mfg Technol TCM Solid Preparat, Nanchang 330006, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R ChinaFang, Yuanying论文数: 0 引用数: 0 h-index: 0机构: Jiangxi Univ Chinese Med, Natl Engn Res Ctr Mfg Technol TCM Solid Preparat, Nanchang 330006, Peoples R China Jiangxi Univ Chinese Med, Coll Pharm, Nanchang 330004, Peoples R China
- [34] Proteolysis-targeting chimera (PROTAC) delivery system: advancing protein degraders towards clinical translationCHEMICAL SOCIETY REVIEWS, 2022, 51 (13) : 5330 - 5350Chen, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Carbone Canc Ctr, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Wisconsin Ctr NanoBioSyst, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USATandon, Ira论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USAHeelan, William论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USAWang, Yixin论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Carbone Canc Ctr, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Wisconsin Ctr NanoBioSyst, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USATang, Weiping论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USAHu, Quanyin论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Carbone Canc Ctr, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Wisconsin Ctr NanoBioSyst, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Pharmaceut Sci Div, Madison, WI 53705 USA
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- [37] Using proteolysis-targeting chimera technology to reduce navitoclax platelet toxicity and improve its senolytic activityNATURE COMMUNICATIONS, 2020, 11 (01)He, Yonghan论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAZhang, Xuan论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Med Chem, Gainesville, FL 32611 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAChang, Jianhui论文数: 0 引用数: 0 h-index: 0机构: Univ Arkansas Med Sci, Dept Pharmaceut Sci, Little Rock, AR 72205 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA论文数: 引用数: h-index:机构:Zhang, Peiyi论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Med Chem, Gainesville, FL 32611 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAWang, Yingying论文数: 0 引用数: 0 h-index: 0机构: Univ Arkansas Med Sci, Dept Pharmaceut Sci, Little Rock, AR 72205 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAKhan, Sajid论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USALiu, Xingui论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAZhang, Xin论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USALv, Dongwen论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USASong, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Arkansas Med Sci, Dept Pharmaceut Sci, Little Rock, AR 72205 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USALi, Wen论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAThummuri, Dinesh论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAYuan, Yaxia论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAWiegand, Janet S.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAOrtiz, Yuma T.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USABudamagunta, Vivekananda论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAElisseeff, Jennifer H.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sch Med, Translat Tissue Engn Ctr, Wilmer Eye Inst, Baltimore, MD USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USACampisi, Judith论文数: 0 引用数: 0 h-index: 0机构: Buck Inst Res Aging, Novato, CA USA Lawrence Berkeley Natl Lab, Berkeley, CA USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAAlmeida, Maria论文数: 0 引用数: 0 h-index: 0机构: Univ Arkansas Med Sci, Ctr Osteoporosis & Metab Bone Dis, Div Endocrinol & Metab, Little Rock, AR 72205 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAZheng, Guangrong论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Med Chem, Gainesville, FL 32611 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USAZhou, Daohong论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA Univ Florida, Coll Pharm, Dept Pharmacodynam, Gainesville, FL 32610 USA
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