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- [21] Design, synthesis, and biological evaluation of novel BTK-targeting proteolysis targeting chimeras (PROTACs) with enhanced pharmacokinetic propertiesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 289Lin, Ying论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaLiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Peoples Hosp 5, Dept Pharm, 801 Heqing Rd, Shanghai 200240, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaTian, Xinjian论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaWang, Jin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaSu, Huahua论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaXiang, Jianpin论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Jiangsu, Peoples R China Nanjing Univ Chinese Med, State Key Lab Technol Chinese Med Pharmaceut Proc, Nanjing 210023, Jiangsu, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaCao, Tao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Jiangsu, Peoples R China Nanjing Univ Chinese Med, State Key Lab Technol Chinese Med Pharmaceut Proc, Nanjing 210023, Jiangsu, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaWang, Yonghui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaXie, Qiong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaYu, Xufen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Key Lab Smart Drug Delivery, Minist Educ, Shanghai 201203, Peoples R China Fudan Univ, MOE Innovat Ctr New Drug Dev Immune Inflammatory D, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China
- [22] Discovery and biological evaluation of proteolysis targeting chimeras (PROTACs) as an EGFR degraders based on osimertinib and lenalidomideBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 30 (12)He, Kailun论文数: 0 引用数: 0 h-index: 0机构: Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R ChinaZhang, Zhuo论文数: 0 引用数: 0 h-index: 0机构: Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R ChinaWang, Wenbing论文数: 0 引用数: 0 h-index: 0机构: Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R ChinaZheng, Xiaoliang论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Acad Med Sci, Ctr Mol Med, Hangzhou 310032, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R ChinaWang, Xiaoju论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Acad Med Sci, Ctr Mol Med, Hangzhou 310032, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R ChinaZhang, Xingxian论文数: 0 引用数: 0 h-index: 0机构: Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China Zhejicmg Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China
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- [24] Design, Synthesis, and Biological Evaluation of Novel EGFR PROTACs Targeting C797S MutationJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (09) : 7283 - 7300Zhu, Yasheng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYe, Xiuquan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWu, Yuxing论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaShen, Hao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaCai, Zeyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaXia, Fei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaMin, Wenjian论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaHou, Yi论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWang, Liping论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWang, Xiao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaXiao, Yibei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, Chongqing Innovat Inst, Chongqing 401135, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYang, Peng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Inst Innovat Drug Discovery & Dev, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China
- [25] Design, synthesis and biological evaluation of Proteolysis Targeting Chimeras (PROTACs) as a BTK degraders with improved pharmacokinetic propertiesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 30 (03)Jaime-Figueroa, Saul论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USABuhimschi, Alexandru D.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USAToure, Momar论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USAHines, John论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USACrews, Craig M.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA Yale Univ, Dept Chem, New Haven, CT 06520 USA Yale Sch Med, Dept Pharmacol, New Haven, CT 06510 USA Yale Univ, Dept Mol Cellular & Dev Biol, New Haven, CT 06511 USA
- [26] Synthesis and biological evaluation of D-amino acid oxidase inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (12) : 3357 - 3359Ferraris, Dana论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USADuvall, Bridget论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USAKo, Yao-Sen论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USAThomas, Ajit G.论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USARojas, Camilo论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USAMajer, Pavel论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USAHashimoto, Kenji论文数: 0 引用数: 0 h-index: 0机构: Chiba Univ Ctr Forens Mental Hlth, Div Clin Neurosci, Chiba 2608670, Japan MGI Pharma Inc, Baltimore, MD 21224 USATsukamoto, Takashi论文数: 0 引用数: 0 h-index: 0机构: MGI Pharma Inc, Baltimore, MD 21224 USA MGI Pharma Inc, Baltimore, MD 21224 USA
- [27] Phenol-Benzoxazolone bioisosteres: Synthesis and biological evaluation of tricyclic GluN2B-selective N-methyl- d-aspartate receptor antagonistsARCHIV DER PHARMAZIE, 2022, 355 (09)Markus, Alexander论文数: 0 引用数: 0 h-index: 0机构: Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanySchreiber, Julian A.论文数: 0 引用数: 0 h-index: 0机构: Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany Univ Hosp Munster, Inst Genet Heart Dis IfGH, Dept Cardiovasc Med Cellular Electrophysiol & Mol, Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanyGoerges, Gunnar论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Munster, Inst Genet Heart Dis IfGH, Dept Cardiovasc Med Cellular Electrophysiol & Mol, Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanyFrehland, Bastian论文数: 0 引用数: 0 h-index: 0机构: Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanySeebohm, Guiscard论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Munster, Inst Genet Heart Dis IfGH, Dept Cardiovasc Med Cellular Electrophysiol & Mol, Munster, Germany Westfalische Wilhelms Univ Munster, Chem Biol Ion Channels Chembion, GRK 2515, Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanySchepmann, Dirk论文数: 0 引用数: 0 h-index: 0机构: Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, GermanyWuensch, Bernhard论文数: 0 引用数: 0 h-index: 0机构: Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany Westfalische Wilhelms Univ Munster, Chem Biol Ion Channels Chembion, GRK 2515, Munster, Germany Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany
- [28] Design, Synthesis, and Biological Evaluation of Proteolysis Targeting Chimeras (PROTACs) for the Dual Degradation of IGF-1R and SrcMOLECULES, 2020, 25 (08):Manda, Sudhakar论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South KoreaLee, Na Keum论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South KoreaOh, Dong-Chan论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Coll Pharm, Inst Nat Prod Res, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South KoreaLee, Jeeyeon论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Coll Pharm, 1 Gwanak Ro, Seoul 08826, South Korea
- [29] In-silico Screening and Synthesis of Benzo[c]Pyridazines Targeting N-Methyl D-Aspartate Glutamate Receptor for the Treatment of SeizuresCHEMISTRY & BIODIVERSITY, 2025, 22 (02)Mishra, Prem Shankar论文数: 0 引用数: 0 h-index: 0机构: Galgotias Univ, Sch Med & Allied Sci, Greater Noida 203201, India Galgotias Univ, Sch Med & Allied Sci, Greater Noida 203201, IndiaMishra, Rakhi论文数: 0 引用数: 0 h-index: 0机构: Noida Inst Engn & Technol, Pharm Inst, Greater Noida 201306, Uttar Pradesh, India Galgotias Univ, Sch Med & Allied Sci, Greater Noida 203201, IndiaMalik, Abdul论文数: 0 引用数: 0 h-index: 0机构: King Saud Univ, Coll Pharm, Dept Pharmaceut, Riyadh 11451, Saudi Arabia Galgotias Univ, Sch Med & Allied Sci, Greater Noida 203201, IndiaKhan, Azmat Ali论文数: 0 引用数: 0 h-index: 0机构: King Saud Univ, Coll Pharm, Dept Pharmaceut Chem, Pharmaceut Biotechnol Lab, Riyadh 11451, Saudi Arabia Galgotias Univ, Sch Med & Allied Sci, Greater Noida 203201, India
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