Overcoming clinical BCR-ABL1 compound mutant resistance with combined ponatinib and asciminib therapy

被引:2
|
作者
Eide, Christopher A. [1 ]
Brewer, Diana [1 ]
Xie, Tao [2 ]
Schultz, Anna Reister [1 ]
Savage, Samantha L. [1 ]
Muratcioglu, Serena [3 ]
Merz, Noah [1 ]
Press, Richard D. [4 ]
O'Hare, Thomas [5 ]
Jacob, Thomas [6 ]
Vu, Tania Q. [6 ,7 ]
Tognon, Cristina E. [1 ]
Macey, Tara A. [1 ]
Kuriyan, John [3 ,8 ]
Kalodimos, Charalampos G. [2 ]
Druker, Brian J. [1 ]
机构
[1] Oregon Hlth & Sci Univ, Knight Canc Inst, Div Hematol & Med Oncol, Portland, OR 97239 USA
[2] St Jude Childrens Res Hosp, Dept Struct Biol, Memphis, TN USA
[3] Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN USA
[4] Oregon Hlth & Sci Univ, Knight Canc Inst, Dept Pathol, Portland, OR USA
[5] Univ Utah, Huntsman Canc Inst, Div Hematol & Hematol Malignancies, Salt Lake City, UT USA
[6] Oregon Hlth & Sci Univ, Dept Biomed Engn, Portland, OR USA
[7] Oregon Hlth & Sci Univ, Ctr Spatial Syst Biosci, Portland, OR USA
[8] Vanderbilt Coll Arts & Sci, Dept Chem, Nashville, TN USA
关键词
PROTEIN;
D O I
10.1016/j.ccell.2024.08.004
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:1486 / 1488
页数:3
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