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- [41] Targeting PI3Kα overcomes resistance to KRasG12C inhibitors mediated by activation of EGFR and/or IGF1RACTA PHARMACOLOGICA SINICA, 2023, 44 (05) : 1083 - 1094Qi, Wei-liang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Nanchang Univ, Coll Pharm, 461 Bayi Rd, Nanchang 330006, Jiangxi, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaLi, Hui-yu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaWang, Yi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaXu, Lan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaDeng, Jie-ting论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaZhang, Xi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaWang, Yu-xiang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R ChinaMeng, Ling-hua论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, 501 Haike Rd, Shanghai 201203, Peoples R China
- [42] Targeting PI3Kα overcomes resistance to KRasG12C inhibitors mediated by activation of EGFR and/or IGF1RActa Pharmacologica Sinica, 2023, 44 : 1083 - 1094Wei-liang Qi论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiHui-yu Li论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiYi Wang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiLan Xu论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiJie-ting Deng论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiXi Zhang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiYu-xiang Wang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of AntiLing-hua Meng论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Division of Anti
- [43] KRASG12c-Mutant NSCLC Under Targeted Therapy in China: Lessons from Eight CasesJOURNAL OF THORACIC ONCOLOGY, 2024, 19 (10) : S649 - S649Li, Y.论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R China Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R ChinaDai, M.论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R China Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R ChinaZhang, R.论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R China Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R ChinaNie, X.论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R China Huazhong Univ Sci & Technol, Tongji Med Coll, Union Hosp, Wuhan 430022, Hubei, Peoples R China
- [44] Combination RASG12C(ON) and RASMULTI(ON) inhibition overcomes resistance and prolongs durability in preclinical models of mutant KRASG12C-driven cancersCANCER RESEARCH, 2024, 84 (06)Wei, Xing论文数: 0 引用数: 0 h-index: 0Holderfield, Matthew论文数: 0 引用数: 0 h-index: 0Yang, Yu Chi论文数: 0 引用数: 0 h-index: 0Seamon, Kyle论文数: 0 引用数: 0 h-index: 0Dinglasan, Jay论文数: 0 引用数: 0 h-index: 0Montazar, Nilufar论文数: 0 引用数: 0 h-index: 0Lee, Bianca论文数: 0 引用数: 0 h-index: 0Cai, Shurui论文数: 0 引用数: 0 h-index: 0Lai, Lick论文数: 0 引用数: 0 h-index: 0Aronchik, Ida论文数: 0 引用数: 0 h-index: 0Chang, Stephanie论文数: 0 引用数: 0 h-index: 0Wang, Zhican论文数: 0 引用数: 0 h-index: 0Wildes, Pete论文数: 0 引用数: 0 h-index: 0Smith, Jacqueline A.论文数: 0 引用数: 0 h-index: 0Jiang, Jingjing论文数: 0 引用数: 0 h-index: 0Singh, Mallika论文数: 0 引用数: 0 h-index: 0
- [45] Co-targeting SOS1 enhances the antitumor effects of KRASG12C inhibitors by addressing intrinsic and acquired resistanceNATURE CANCER, 2024, 5 (09) : 1352 - 1370Thatikonda, Venu论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Exscientia, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaLyu, Hengyu论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaJurado, Sabine论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaKostyrko, Kaja论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaBristow, Christopher A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaAlbrecht, Christoph论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaAlpar, Donat论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaArnhof, Heribert论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaBergner, Oliver论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaBosch, Karin论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaFeng, Ningping论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaGao, Sisi论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaGerlach, Daniel论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaGmachl, Michael论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaHinkel, Melanie论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaLieb, Simone论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaJeschko, Astrid论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaMachado, Annette A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaMadensky, Thomas论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaMarszalek, Ethan D.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaMahendra, Mikhila论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaMelo-Zainzinger, Gabriella论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaMolkentine, Jessica M.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaJaeger, Philipp A.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaPeng, David H.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaSchenk, Robyn L.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaSorokin, Alexey论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Gastrointestinal Med Oncol, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaStrauss, Sandra论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaTrapani, Francesca论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaKopetz, Scott论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Gastrointestinal Med Oncol, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaVellano, Christopher P.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaPetronczki, Mark论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaKraut, Norbert论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaHeffernan, Timothy P.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaMarszalek, Joseph R.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Therapeut Discovery Div, Translat Res Adv Therapeut & Innovat Oncol TRACTIO, Houston, TX USA Boehringer Ingelheim RCV, Vienna, AustriaPearson, Mark论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaWaizenegger, Irene C.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, AustriaHofmann, Marco H.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV, Vienna, Austria Boehringer Ingelheim RCV, Vienna, Austria
- [46] High EGFR Expression Confers Acquired Resistance to Adagrasib - In Vitro Study Using KRASg12C Mutated Lung Cancer CellsJOURNAL OF THORACIC ONCOLOGY, 2024, 19 (10) : S315 - S315Hamada, A.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanSuda, K.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanObata, K.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanSato, H.论文数: 0 引用数: 0 h-index: 0机构: Yamagata Univ, Well Being Inst, Yamagata, Japan Kindai Univ, Fac Med, Osaka, JapanOiki, H.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanFukuda, S.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, Japan论文数: 引用数: h-index:机构:Ito, M.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanSoh, J.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanTsutani, Y.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, JapanMitsudomi, T.论文数: 0 引用数: 0 h-index: 0机构: Kindai Univ, Fac Med, Osaka, Japan Kindai Univ, Fac Med, Osaka, Japan
- [47] Phase 2 Trial of Neoadjuvant KRASG12C Directed Therapy with Adagrasib (MRTX849) With or Without Nivolumab in Resectable NSCLC (Neo-KAN)JOURNAL OF THORACIC ONCOLOGY, 2022, 17 (09) : S235 - S235Scott, S. C.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAHu, C.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USASmith, K.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAAnagnostou, V.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USALee, J.论文数: 0 引用数: 0 h-index: 0机构: UCLA Hlth, Los Angeles, CA USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA论文数: 引用数: h-index:机构:Illei, P.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAProphet, E.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USARosner, S.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAEttinger, D.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAFeliciano, J.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAHann, C.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USALam, V.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USALevy, B.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAMurray, J.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USABrahmer, J.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAForde, P.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USAMarrone, K.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA Johns Hopkins Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD USA
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