Design, Synthesis, Antibacterial, and Antifungal Activity Evaluation of Novel Pyrimidine Derivatives Incorporating Amide and 1,3,4-Thiadiazole Thioether Moieties

被引：0
|
作者：
Shuang-Xue Wu [1 ]
Jing Liu [1 ]
Bo-Xi Tan [1 ]
Can He [1 ]
Wen-Qing Wu [1 ]
Lu Yu [1 ]
Pei Li [1 ]
机构：
[1] School of Liquor and Food Engineering,
[2] Guizhou University,undefined
[3] Qiandongnan Engineering and Technology Research Center for Comprehensive Utilization of National Medicine,undefined
[4] Kaili University,undefined
来源：
Russian Journal of General Chemistry | 2024年 / 94卷 / 12期
关键词：
pyrimidine; amide; 1,3,4-thiadiazole thioether; antibacterial activity; antifungal activity;
D O I：
10.1134/S1070363224120375
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：3448 / 3455
页数：7
相关论文
共 50 条
  • [21] Synthesis and Bioactivity Evaluation of Novel Thiochroman-4-One Derivatives Incorporating Carboxamide and 1, 3, 4-Thiadiazole Thioether Moieties
    Yu, Lu
    Xiao, Lingling
    Li, Pei
    Chi, Jiyan
    Li, Jie
    Tan, Shuming
    JOURNAL OF CHEMISTRY, 2022, 2022
  • [22] Synthesis and Antiproliferative Activity of Novel 1,3,4-Thiadiazole Derivatives
    Liu, Tingting
    Wan, Yichao
    Fang, Hao
    CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 36 (02) : 417 - 424
  • [23] Design, Synthesis, and Bioactivity Evaluation of Novel 1,3,4-Thiadiazole Sulfone-Derived Compounds Incorporating an Amide Moiety as Active Antibacterial Agents
    S. Song
    L. Yu
    B. Tan
    J. Liu
    S. Wu
    P. Li
    Russian Journal of General Chemistry, 2024, 94 (10) : 2789 - 2796
  • [24] Novel Flavonol Derivatives Containing 1,3,4-Thiadiazole as Potential Antifungal Agents: Design, Synthesis, and Biological Evaluation
    Zhou, Yuanxiang
    Gong, Chenyu
    Sun, Zhiling
    Zeng, Wei
    Meng, Kaini
    An, Youshan
    Hu, Yuzhi
    Xue, Wei
    ACS OMEGA, 2024,
  • [25] Synthesis and Evaluation of New 1,3,4-Thiadiazole Derivatives as Potent Antifungal Agents
    Karaburun, Ahmet Cagri
    Cevik, Ulviye Acar
    Osmaniye, Derya
    Saglik, Begum Nurpelin
    Cavusoglu, Betul Kaya
    Levent, Serkan
    Ozkay, Yusuf
    Koparal, Ali Savas
    Behcet, Mustafa
    Kaplancikli, Zafer Asim
    MOLECULES, 2018, 23 (12):
  • [26] Synthesis and Antifungal Activity of 1,3,4-Thiadiazole Derivatives Containing Pyridine Group
    Zhang, Lin-Jiong
    Yang, Ming-Yan
    Sun, Zhao-Hui
    Tan, Cheng-Xia
    Weng, Jian-Quan
    Wu, Hong-Ke
    Liu, Xing-Hai
    LETTERS IN DRUG DESIGN & DISCOVERY, 2014, 11 (09) : 1107 - 1111
  • [27] SYNTHESIS OF NOVEL THIAZOLE AND 1,3,4-THIADIAZOLE DERIVATIVES INCORPORATING PHENYLSULFONYL MOIETY
    Mekky, Ahmed E. M.
    Darweesh, Ahmed F.
    Salman, Amani A.
    Farag, Ahmad M.
    HETEROCYCLES, 2014, 89 (08) : 1827 - 1843
  • [28] SYNTHESIS AND ANTIMICROBIAL EVALUATION OF NEW PYRAZOLE, THIOPHENE, THIAZOLE AND 1,3,4-THIADIAZOLE DERIVATIVES INCORPORATING PYRIMIDINE RING
    Farag, Ahmad M.
    Kheder, Nabila A.
    Mabkhot, Yahia N.
    HETEROCYCLES, 2009, 78 (07) : 1787 - 1798
  • [29] STUDIES ON 1,3,4-THIADIAZOLE DERIVATIVES .8. ANTIBACTERIAL ACTIVITIES OF 1,3,4-THIADIAZOLE DERIVATIVES
    OHTA, M
    OYA, H
    MIFUNE, A
    YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 1953, 73 (08): : 852 - 854
  • [30] Synthesis and cytotoxic evaluation of new colchicine derivatives bearing 1,3,4-thiadiazole moieties
    Shen, Li-Hong
    Li, Hong-Yu
    Shang, Hui-Xia
    Tian, Shu-Ting
    Lai, Yi-Sheng
    Liu, Li-Jie
    CHINESE CHEMICAL LETTERS, 2013, 24 (04) : 299 - 302
12345