Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols

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作者
Strauss, Michael J. [1 ]
Liu, Kaylee X. [1 ,2 ]
Greaves, Megan E. [1 ]
Dahl, Jakob C. [1 ,3 ]
Kim, Seoung-Tae [1 ]
Wu, Yong-Jin [4 ]
Schmidt, Michael A. [5 ]
Scola, Paul M. [4 ]
Buchwald, Stephen L. [1 ]
机构
[1] Department of Chemistry, Massachusetts Institute of Technology, 77 Massachusetts Ave, Cambridge,MA,02139, United States
[2] Department of Chemistry, Wellesley College, 106 Central St, Wellesley,MA,02481, United States
[3] Department of Chemical Engineering, Massachusetts Institute of Technology, 77 Massachusetts Ave, Cambridge,MA,02139, United States
[4] Department of Discovery Chemistry, Bristol Myers Squibb, 250 Water St, Cambridge,MA,02141, United States
[5] Chemical Process Development, Bristol Myers Squibb, 1 Squibb Dr, New Brunswick,NJ,08901, United States
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61
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页码:18616 / 18625
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