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- [21] Design, synthesis, and biological activity of classical N-[2-amino-4-substituted[(pyrrolo[2,3-D]pyrimidine-5-yl) ethyl]benzoyl)-L-glutamic acids as dual inhibitors of dihydrofolate reductase and thymidylate synthase. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U29 - U29
- [22] ANALOGS OF BIOLOGICAL ACTIVE COMPOUNDS .2. SYNTHESIS OF N-[4-(3-OXO-6-AMINO-2,3-DIHYDRO-1,2,4-BENZOTRIAZIN-2-YL)BENZOYL]-L-GLUTAMIC ACID PHARMAZIE, 1988, 43 (12): : 864 - 864
- [25] SYNTHESIS OF A NOVEL 5-DEAZA-5-THIA ANALOG OF TETRAHYDROFOLIC ACID, N-(P-([(2-AMINO-6,7-DIHYDRO-4-OXO-3H,8H-PYRIMIDO[5,4-B][1,4]THIAZIN-6-YL)METHYL]AMINO)BENZOYL)GLUTAMIC ACID JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1994, (07): : 833 - 836
- [26] Design, synthesis, and biological activities of classical N-{4-[2-(2-amino-4-ethylpyrrolo[2,3-d]pyrimidin-5-yl)ethylbenzoyl}-L-glutamic acid and its 6-methyl derivative as potential dual inhibitors of thymidylate synthase and dihydrofolate reductase and as potential antitumor agents JOURNAL OF MEDICINAL CHEMISTRY, 2003, 46 (04) : 591 - 600