共 50 条
- [1] A comprehensive comparative study on LSD1 in different cancers and tumor specific LSD1 inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 240Dong, Jianshu论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China论文数: 引用数: h-index:机构:Tayyab, Bilal论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLi, Die论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaKang, Lei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaZhang, Huimin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaGong, Huimin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaMa, Xinli论文数: 0 引用数: 0 h-index: 0机构: China US Henan Hormel Canc Inst, 127,Dongming Rd,Jinshui Dist, Zhengzhou 450008, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLi, Jian论文数: 0 引用数: 0 h-index: 0机构: China US Henan Hormel Canc Inst, 127,Dongming Rd,Jinshui Dist, Zhengzhou 450008, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaAgboyibor, Clement论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaBi, Yuefeng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, 100 Kexue Dadao,Gaoxin Dist, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, 100 Kexue Dadao,Gaoxin Dist, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China
- [2] Reversible Lysine Specific Demethylase 1 (LSD1) Inhibitors: A Promising Wrench to Impair LSD1JOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (05) : 2466 - 2488Dai, Xing-Jie论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaLiu, Ying论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaXue, Lei-Peng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaXiong, Xiao-Peng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaZhou, Ying论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaZheng, Yi-Chao论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaLiu, Hong-Min论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China
- [3] Taking LSD1 to a new highCELL, 2005, 122 (05) : 654 - 658Wysocka, J论文数: 0 引用数: 0 h-index: 0机构: Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USA Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USAMilne, TA论文数: 0 引用数: 0 h-index: 0机构: Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USA Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USAAllis, CD论文数: 0 引用数: 0 h-index: 0机构: Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USA Rockefeller Univ, Lab Chromatin Biol, New York, NY 10021 USA
- [4] LSD1 tunes adipose tissuesNature Reviews Molecular Cell Biology, 2014, 15 (7) : 430 - 430Andrea Du Toit论文数: 0 引用数: 0 h-index: 0
- [5] Inhibition of LSD1 for the treatment of cancerCANCER RESEARCH, 2015, 75Smitheman, Kimberly论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USACusan, Monica论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA GlaxoSmithKline, Collegeville, PA USALiu, Yan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAButticello, Michael论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAPappalardi, Melissa论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAFoley, James论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAFederowicz, Kelly论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAVan Aller, Glenn论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAKasparec, Jiri论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USATian, Xinrong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USASuarez, Dominic论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USASchneck, Jess论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USACarson, Jeff论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAMcDevitt, Patrick论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAHo, Thau论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAMcHugh, Charles论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAMiller, William论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAArmstrong, Scott论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA GlaxoSmithKline, Collegeville, PA USAHann, Christine论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Baltimore, MD USA GlaxoSmithKline, Collegeville, PA USAJohnson, Neil论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAKruger, Ryan G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAMohammad, Helai P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAKamat, Shekhar论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Baltimore, MD USA GlaxoSmithKline, Collegeville, PA USA
- [6] LSD1 modulation by allosteric ligandsCANCER RESEARCH, 2019, 79 (13)Emond, Wei B.论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenGeitmann, Matthis论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenJarvius, Malin论文数: 0 引用数: 0 h-index: 0机构: SciLifeLab Drug Discovery & Dev, Uppsala, Sweden Beactica AB, Uppsala, SwedenKoehler, Konrad论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenKallblad, Per论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenNiklasson, Mia论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Uppsala, Sweden Beactica AB, Uppsala, SwedenParrow, Vendela论文数: 0 引用数: 0 h-index: 0机构: SciLifeLab Drug Discovery & Dev, Uppsala, Sweden Beactica AB, Uppsala, SwedenSawant, Rajiv论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenSjoberg, Maria论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, SwedenWinquist, Johan论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, Sweden论文数: 引用数: h-index:机构:Bremberg, Ulf论文数: 0 引用数: 0 h-index: 0机构: Beactica AB, Uppsala, Sweden Beactica AB, Uppsala, Sweden
- [7] Potentiation of immunotherapy by LSD1 modulationCANCER RESEARCH, 2023, 83 (07)Emond, Wei B.论文数: 0 引用数: 0 h-index: 0Sawant, Rajiv论文数: 0 引用数: 0 h-index: 0Geitmann, Matthis论文数: 0 引用数: 0 h-index: 0Winquist, Johan论文数: 0 引用数: 0 h-index: 0Brandt, Peter论文数: 0 引用数: 0 h-index: 0Bremberg, Ulf论文数: 0 引用数: 0 h-index: 0Kallblad, Per论文数: 0 引用数: 0 h-index: 0Parrow, Vendela论文数: 0 引用数: 0 h-index: 0Andersson, Claes论文数: 0 引用数: 0 h-index: 0Blom, Kristin论文数: 0 引用数: 0 h-index: 0Najafi, Nasrin论文数: 0 引用数: 0 h-index: 0Bergstrom, Tobias论文数: 0 引用数: 0 h-index: 0Swartling, Fredrik J.论文数: 0 引用数: 0 h-index: 0Hellstrom, Mats论文数: 0 引用数: 0 h-index: 0Koehler, Konrad F.论文数: 0 引用数: 0 h-index: 0
- [8] Discovery of reversible LSD1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 254Kanouni, Toufike论文数: 0 引用数: 0 h-index: 0机构: Celgene, Chem, San Diego, CA USA Celgene, Chem, San Diego, CA USA
- [9] LSD1 Makes Fat ColorfulTRENDS IN ENDOCRINOLOGY AND METABOLISM, 2017, 28 (01): : 1 - 2Straub, Leon G.论文数: 0 引用数: 0 h-index: 0机构: Swiss Fed Inst Technol, Inst Food Nutr & Hlth, Eidgenoss Tech Hsch, Schorenstr 16, CH-8603 Schwerzenbach, Switzerland Swiss Fed Inst Technol, Inst Food Nutr & Hlth, Eidgenoss Tech Hsch, Schorenstr 16, CH-8603 Schwerzenbach, SwitzerlandWolfrum, Christian论文数: 0 引用数: 0 h-index: 0机构: Swiss Fed Inst Technol, Inst Food Nutr & Hlth, Eidgenoss Tech Hsch, Schorenstr 16, CH-8603 Schwerzenbach, Switzerland Swiss Fed Inst Technol, Inst Food Nutr & Hlth, Eidgenoss Tech Hsch, Schorenstr 16, CH-8603 Schwerzenbach, Switzerland
- [10] The lasting influence of LSD1 in the bloodELIFE, 2013, 2Dent, Sharon Y. R.论文数: 0 引用数: 0 h-index: 0机构: MD Anderson Canc Ctr, Dept Mol Carcinogenesis, Houston, TX 77030 USA MD Anderson Canc Ctr, Dept Mol Carcinogenesis, Houston, TX 77030 USAChandra, Joya论文数: 0 引用数: 0 h-index: 0机构: MD Anderson Canc Ctr, Dept Mol Carcinogenesis, Houston, TX 77030 USA MD Anderson Canc Ctr, Dept Pediat Res, Houston, TX USA MD Anderson Canc Ctr, Dept Mol Carcinogenesis, Houston, TX 77030 USA