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- [1] First-in-human phase I study of the ALK inhibitor LDK378 in advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2012, 30 (15)Mehra, Ranee论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USACamidge, D. Ross论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USASharma, Sunil论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USAFelip, Enriqueta论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USATan, Daniel Shao-Weng论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USAVansteenkiste, Johan F.论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USADe Pas, Tommaso Martino论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USAKim, Dong-Wan论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USASantoro, Armando论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USALiu, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USAGoldwasser, Meredith论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USADai, David论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USARadona, Marietta论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USABoral, Anthony论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USAShaw, Alice Tsang论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Philadelphia, PA 19111 USA
- [2] First-in-human phase 1 study of DS-1062a in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2019, 37 (15)Sands, Jacob M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAShimizu, Toshio论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGaron, Edward B.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGreenberg, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGuevara, Ferdinand M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAHeist, Rebecca Suk论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAKobayashi, Fumiaki论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USANoguchi, Yutaka论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAOkajima, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USATajima, Naoyuki论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USASpira, Alexander I.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAYamamoto, Noboru论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USALisberg, Aaron Elliott论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA
- [3] Phase 1 first-in-human trial of MTB-9655, the first oral inhibitor of ACSS2, in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2022, 40 (16)Perets, Ruth论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelGeva, Ravit论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelMcKean, Meredith论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelGoutopoulos, Andreas论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelErez, Omri论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelPhadnis, Monica论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelYoussoufian, Hagop论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelSchwartz, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelKansra, Vikram论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, IsraelFattaey, Ali论文数: 0 引用数: 0 h-index: 0机构: Rambam Hlth Care Campus, Haifa, Israel
- [4] First-in-human phase I study of an oral HSP9O inhibitor, TAS-116, in advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2017, 35Yanagitani, Noriko论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanHoriike, Atsushi论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanKitazono, Satoru论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanOhyanagi, Fumiyoshi论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanKondo, Shunsuke论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanShimomura, Akihiko论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanFujiwara, Yutaka论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanDoi, Toshihiko论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanKuboki, Yasutoshi论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanKawazoe, Akihito论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanShitara, Kohei论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanOhno, Izumi论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanBanerji, Udai论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanSundar, Raghav论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanOhkubo, Shuichi论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanHuang, Jerry M.论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanNishio, Makoto论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, JapanYamamot, Noboru论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, Japan
- [5] First-in-human study of TAS-115, a novel oral MET/VEGFR inhibitor, in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Matsubara, Nobuaki论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanShitara, Kohei论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanNaito, Yoichi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanKuboki, Yasutoshi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanOhno, Izumi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanTakahashi, Hideaki论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanBando, Hideaki论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanKojima, Takashi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanFuse, Nozomu论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanYamazaki, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanHirayama, Naoki论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanFujita, Hidenori论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanNishida, Toshirou论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, JapanDoi, Toshihiko论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Chiba, Japan
- [6] First-in-human dose escalation study of oral ONC201 in advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Stein, Mark N.论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAMayer, Tina M.论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAMoss, Rebecca Anne论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USASilk, Ann W.论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAChan, Nancy论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAHaffty, Bruce George论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USADiPaola, Robert S.论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USABeckett, Yasmeen论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USABentlyewski, Edward论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAZheng, Ling论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAFang, Bruno论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAAllen, Joshua论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USAMehnert, Janice M.论文数: 0 引用数: 0 h-index: 0机构: Rutgers Canc Inst New Jersey, New Brunswick, NJ USA
- [7] First-in-human phase I study of a selective VEGFR/FGFR dual inhibitor sulfatinib in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2012, 30 (15)Xu, Jian-Ming论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaWang, Yan论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaShen, Lin论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaGong, Jifang论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaHuang, Cheng论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaYe, Chen Yang论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaYang, Li论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaSai, Yang论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R ChinaMu, Hua论文数: 0 引用数: 0 h-index: 0机构: Acad Mil Med Sci, Hosp 307, Ctr Canc, Beijing, Peoples R China
- [8] A first-in-human phase 1 study of a novel PARP7 inhibitor RBN-2397 in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2021, 39 (15)Falchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAPatel, Manish R.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAYap, Timothy A.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAMcEachern, Kristen论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAKuplast-Barr, Kristy论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAUtley, Luke论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USACleary, Lisa论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAManyak, Erika论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USABozon, Viviana论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAParasuraman, Sudha论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USAJohnson, Melissa Lynne论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USA
- [9] First-in-human phase 1 study of pimicotinib (ABSK021), a CSF-1R inhibitor, in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2023, 41 (16)Falchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USALiang, Yan论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAHarvey, R. Donald论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAFu, Siqing论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAWeitao, Yao论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAQin, Yan-Ru论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAZhang, Xiaojing论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAHenry, Jason Timothy论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAZou, Qingping论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAShan, Boyao论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USALiang, Pan论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAWang, Chen论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USALi, Wenjia论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAPamuklar, Zehra Nurgul论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAPei, Yi论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAChang, Zhiwei论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAWang, Jiaqiang论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAPiha-Paul, Sarina A.论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USABhave, Manali A.论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USAYin, Yongmei论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USA
- [10] First-in-human, first-in-class phase 1 study of a novel oral multi-AGC kinase inhibitor AT13148 in patients (pis) with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Kumar, Rajiv论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandMateo, Joaquin论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandSmith, Alan D.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandKhan, Khurum Hayat论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandRuddle, Ruth论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandSwales, Karen E.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandDecordova, Shaun论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandBackholer, Zoe论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandJones, Paul论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandTran, Christine论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandSeeramraddi, Satyanarayana论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandMcLeod, Robert论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandYap, Timothy Anthony论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandRaynaud, Florence I.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandGarrett, Michelle D.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, EnglandBanerji, Udai论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Drug Dev Unit, London SW3 6JB, England