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- [21] Multiple conformational states of the HPK1 kinase domain in complex with sunitinib reveal the structural changes accompanying HPK1 trans-regulationJOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 294 (23) : 9029 - 9036Johnson, Eric论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAMcTigue, Michele论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAGallego, Rebecca A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAJohnson, Ted W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USATimofeevski, Sergei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAMaestre, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAFisher, Timothy S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USAKania, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USASawasdikosol, Sansana论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USABurakoff, Steven论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USACronin, Ciaran N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, 10770 Sci Ctr Dr,CB2, San Diego, CA 92121 USA
- [22] Discovery of Pyridine-2-Carboxamides Derivatives as Potent and Selective HPK1 Inhibitors for the Treatment of CancerJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (23) : 21520 - 21544Peng, Jingjing论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaDing, Xiaoyu论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaChen, Celia Xiaojing论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaZhao, Pei论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaDing, Xiao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaZhang, Man论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaAliper, Alex论文数: 0 引用数: 0 h-index: 0机构: Insil Med AI Ltd, Abu Dhabi 145748, U Arab Emirates Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaRen, Feng论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaLu, Hongfu论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaZhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med AI Ltd, Abu Dhabi 145748, U Arab Emirates Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China
- [23] Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors as Preclinical Immunotherapy Tool CompoundsACS MEDICINAL CHEMISTRY LETTERS, 2021, 12 (04): : 653 - 661Vara, Brandon A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALevi, Samuel M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAAchab, Abdelghani论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USACandito, David A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAFradera, Xavier论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Computat & Struct Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALesburg, Charles A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Computat & Struct Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAKawamura, Shuhei论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALacey, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALim, Jongwon论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAMethot, Joey L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAXu, Zangwei论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAXu, Haiyan论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USASmith, Dustin M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Pharmacokinet & Drug Metab, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAPiesvaux, Jennifer A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAMiller, J. Richard论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USABittinger, Mark论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Oncol Early Discovery, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USARanganath, Sheila H.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Oncol Early Discovery, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USABennett, David J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USADiMauro, Erin F.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAPasternak, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA
- [24] Development and characterization of small molecule HPK1 inhibitors.CANCER RESEARCH, 2021, 81 (13)Kujawa, Maciej论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandZimolag, Eliza论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGalezowski, Michal论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGuzik, Pawel论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandDudek, Agata论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGondela, Andrzej论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandNowogrodzki, Marcin论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGirardi, Marianna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandKrolenko, Kostiantyn论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBugaj, Marta论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSudol, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGibas, Agnieszka论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSzeremeta-Spisak, Joanna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBobowska, Aneta论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandZastawna, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandWyrebek, Przemyslaw论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBoutard, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandWieckowska, Aleksandra论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandJasnosz, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSchonemann, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandZuchowicz, Karol论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSynak, David论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandKulesza, Urszula论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandLeventes, Oleksandr论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSwirski, Mateusz论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandSasmal, Sujit论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandGluza, Karolina论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandKret, Patryk论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandOgorek, Mateusz论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandMichalik, Kinga论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBanaszak, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandPodkowa, Adrian论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandWnuk-Lipinska, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandDobrzanska, Monika论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandLittlewood, Peter论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBrzozka, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandBartosik, Anna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, PolandChmielewski, Stefan论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut, Krakow, Poland Ryvu Therapeut, Krakow, Poland
- [25] Discovery and Optimization of Pyrazine Carboxamide AZ3246, a Selective HPK1 InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (04) : 4582 - 4595Shields, Jason D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandBaker, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandBalazs, Amber Y. S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandBommakanti, Gayathri论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandCasella, Robert论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Adv Drug Delivery, Pharmaceut Sci, R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandCao, Shenggen论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, Beijing 100176, Peoples R China AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandCook, Steve论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Adv Drug Delivery, Pharmaceut Sci, R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandEscobar, Randolph A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandFawell, Stephen论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandGibbons, Francis D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandGiblin, Kathryn A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandGoldberg, Frederick W.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandGosselin, Eric论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandGrebe, Tyler论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandHariparsad, Niresh论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandHatoum-Mokdad, Holia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandHowells, Rachel论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandHughes, Samantha J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandJackson, Anne论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandReddy, Iswarya Karapa论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandKettle, Jason G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandLamont, Gillian M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandLamont, Scott论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Early Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandLi, Min论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, Beijing 100176, Peoples R China AstraZeneca, Discovery Sci, R&D, Cambridge CB2 0AA, EnglandLill, Sten O. 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