共 50 条
- [1] Discovery of GNE-6893, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of HPK1ACS MEDICINAL CHEMISTRY LETTERS, 2024, 15 (09): : 1606 - 1614Tellis, John C.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAWei, BinQing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASiu, Michael论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAAn, Le论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChan, Grace Kayan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChen, Yong论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Inc, Beijing 100176, Peoples R China Genentech Inc, South San Francisco, CA 94080 USADu, Xiangnan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAGazzard, Lewis论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAHu, Baihua论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Inc, Beijing 100176, Peoples R China Genentech Inc, South San Francisco, CA 94080 USAKiefer, James论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAKakiuchi-Kiyota, Satoko论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USALainchbury, Michael论文数: 0 引用数: 0 h-index: 0机构: Charles River Labs, Harlow CM19 5TR, Essex, England Genentech Inc, South San Francisco, CA 94080 USALinehan, Jonathan L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USALuo, Xifeng论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Inc, Beijing 100176, Peoples R China Genentech Inc, South San Francisco, CA 94080 USAMalhotra, Sushant论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAMendonca, Rohan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USARan, Yinqing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASethuraman, Vijay论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASeward, Eileen论文数: 0 引用数: 0 h-index: 0机构: Charles River Labs, Harlow CM19 5TR, Essex, England Genentech Inc, South San Francisco, CA 94080 USASneeringer, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASu, Dian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAWu, Ping论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAMoffat, John G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAHeffron, Timothy P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChoo, Edna F.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChan, Bryan K.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USA
- [2] Discovery of novel, potent, selective and orally bioavailable HPK1 inhibitor for enhancing the efficacy of anti-PD-L1 antibodyEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 267Zeng, Shenxin论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaWu, Mingfei论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Hangzhou Inst Innovat Med, Inst Drug Discovery & Design, Coll Pharmaceut Sci, Hangzhou 310058, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaJin, Yuyuan论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaYe, Yingqiao论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaXia, Heye论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaChen, Xinyi论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaChe, Jinxin论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Hangzhou Inst Innovat Med, Inst Drug Discovery & Design, Coll Pharmaceut Sci, Hangzhou 310058, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaWang, Zunyuan论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaWu, Ying论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaDong, Xiaowu论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Hangzhou Inst Innovat Med, Inst Drug Discovery & Design, Coll Pharmaceut Sci, Hangzhou 310058, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaChen, Yinqiao论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R ChinaHuang, Wenhai论文数: 0 引用数: 0 h-index: 0机构: Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Sch Pharm, Key Lab Neuropsychiat Drug Res Zhejiang Prov, Hangzhou 311399, Zhejiang, Peoples R China Hangzhou Med Coll, Key Discipline Zhejiang Prov Publ Hlth & Prevent M, Class 1, Category A, Hangzhou, Peoples R China Hangzhou Med Coll, Affiliated Yongkang Peoples Hosp 1, Sch Pharmaceut Sci, Hangzhou 311399, Zhejiang, Peoples R China
- [3] Discovery of Pyrazolopyridine Derivatives as HPK1 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2023, 14 (01): : 5 - 10Ye, Qinda论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USALiu, Kai论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAYe, Hai-Fen论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAPan, Jun论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USASokolsky, Alexander论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAWang, Anlai论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAZhang, Ke论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAHummel, Joshua R.论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAKong, Ling论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USABehshad, Elham论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAHe, Xin论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAConlen, Patricia论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAStump, Kristine论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAYe, Min论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USADiamond, Sharon论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAYeleswaram, Swamy论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAAtasoylu, Onur论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAVechorkin, Oleg论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE 19803 USA Incyte Res Inst, Wilmington, DE 19803 USA
- [4] Discovery of Novel PROTAC-Based HPK1 Degraders with High Potency and Selectivity for Cancer ImmunotherapyJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (21) : 18682 - 18698Zhang, Zhimin论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaGuo, Liubin论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhao, Mengting论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaPan, Hao论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaDong, Zhao论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaWang, Ling论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaYang, Xi论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhang, Zhiping论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaWu, Mengqiang论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaChang, Yujie论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaYang, Yacheng论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaSun, Linan论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaLiu, Sirui论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhu, Rongyao论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZheng, Haowen论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaDai, Xinyu论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhang, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaJiang, Chunhua论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhu, Zhuangzhi论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaZhang, Yuchen论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R ChinaLiu, Dongzhou论文数: 0 引用数: 0 h-index: 0机构: Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China Huadong Med, Global Drug R&D Ctr, Hangzhou 310011, Peoples R China
- [5] HPK1 kinase inhibitor: a sufficient approach to target HPK1 to modulate T cell activation in cancer immunotherapy compared with degradersFRONTIERS IN IMMUNOLOGY, 2025, 16Wang, Qin论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaZhu, Xinyi论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaLi, Jing论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Med Chem, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaXu, Sanjia论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Med Chem, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaWang, Ali论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaZhang, Xinwen论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaWang, Xingxing论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Med Chem, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaCai, Xiaopeng论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Med Chem, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaXing, Haimei论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaLiu, Ye论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaLiu, Xuesong论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaWang, Zhiwei论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Med Chem, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaWang, Lai论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Res & Clin Dev, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R ChinaYuan, Xi论文数: 0 引用数: 0 h-index: 0机构: BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China BeiGene Beijing Co Ltd, Dept Biol, Beijing, Peoples R China
- [6] HPK1 as a novel target for cancer immunotherapyIMMUNOLOGIC RESEARCH, 2012, 54 (1-3) : 262 - 265Sawasdikosol, Sansana论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USAZha, Renyuan论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USAYang, Boyu论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USABurakoff, Steven论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Mt Sinai Sch Med, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA
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- [8] Identification of Potent Reverse Indazole Inhibitors for HPK1ACS MEDICINAL CHEMISTRY LETTERS, 2021, 12 (03): : 459 - 466Yu, Elsie C.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAMethot, Joey L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAFradera, Xavier论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Computat & Struct Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALesburg, Charles A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Computat & Struct Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALacey, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USASiliphaivanh, Phieng论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USALiu, Ping论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, External Discovery Chem, Rahway, NJ 07065 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USASmith, Dustin M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Pharmacokinet & Drug Metab, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAXu, Zangwei论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAPiesvaux, Jennifer A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAKawamura, Shuhei论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAXu, Haiyan论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAMiller, J. Richard论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Quantitat Biosci, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USABittinger, Mark论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Oncol Early Discovery, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USAPasternak, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA Merck & Co Inc, Discovery Chem, Boston, MA 02115 USA
- [9] HPK1 as a novel target for cancer immunotherapyImmunologic Research, 2012, 54 : 262 - 265Sansana Sawasdikosol论文数: 0 引用数: 0 h-index: 0机构: Mount Sinai School of Medicine,Department of Oncological Sciences, Tisch Cancer InstituteRenyuan Zha论文数: 0 引用数: 0 h-index: 0机构: Mount Sinai School of Medicine,Department of Oncological Sciences, Tisch Cancer InstituteBoyu Yang论文数: 0 引用数: 0 h-index: 0机构: Mount Sinai School of Medicine,Department of Oncological Sciences, Tisch Cancer InstituteSteven Burakoff论文数: 0 引用数: 0 h-index: 0机构: Mount Sinai School of Medicine,Department of Oncological Sciences, Tisch Cancer Institute
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