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- [41] Exploring Targeted Degradation Strategy for Oncogenic KRASG12CCELL CHEMICAL BIOLOGY, 2020, 27 (01): : 19 - +Zeng, Mei论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAXiong, Yuan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USASafaee, Nozhat论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Donovan, Katherine A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAYuan, Christine J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USANabet, Behnam论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGero, Thomas W.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAFeru, Frederic论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USALi, Lianbo论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGondi, Sudershan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAOmbelets, Lincoln J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAQuan, Chunshan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Belfer Ctr Appl Canc Sci, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Scott, David A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAWestover, Kenneth D.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAFischer, Eric S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA
- [42] Hedgehog signalling is involved in acquired resistance to KRASG12C inhibitors in lung cancer cellsCell Death & Disease, 15Chaeyoung Lee论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesJawoon Yi论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesJihwan Park论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesByungyong Ahn论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesYoung-Wook Won论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesJiHeung Jeon论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesByung Ju Lee论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesWha Ja Cho论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological SciencesJeong Woo Park论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Biological Sciences
- [43] KRASG12C inhibition in tumor therapyONKOLOGE, 2021, 27 (01): : 72 - 73Alakus, Hakan论文数: 0 引用数: 0 h-index: 0机构: Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, Germany Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, GermanyHartmann, Milan论文数: 0 引用数: 0 h-index: 0机构: Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, Germany Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, Germany论文数: 引用数: h-index:机构:Bruns, Christiane论文数: 0 引用数: 0 h-index: 0机构: Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, Germany Univ Cologne, Klin & Poliklin Allgemein Viszeral & Tumorchirurg, Univ Klinikum Koln AoR, Kerpener Str 62, D-50937 Cologne, Germany
- [44] Evaluation of KRASG12C inhibitor responses in novel murine KRASG12C lung cancer cell line modelsFRONTIERS IN ONCOLOGY, 2023, 13Sisler, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USA Rocky Mt Reg VA Med Ctr, Eastern Colorado VA Healthcare Syst, Aurora, CO 80045 USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USAHinz, Trista K.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USA Rocky Mt Reg VA Med Ctr, Eastern Colorado VA Healthcare Syst, Aurora, CO 80045 USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USALe, Anh T.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Med, Aurora, CO USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USAKleczko, Emily K.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Med, Aurora, CO USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USANemenoff, Raphael A.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Med, Aurora, CO USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USAHeasley, Lynn E.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USA Rocky Mt Reg VA Med Ctr, Eastern Colorado VA Healthcare Syst, Aurora, CO 80045 USA Univ Colorado Anschutz Med Campus, Dept Craniofacial Biol, Aurora, CO 80045 USA
- [45] Inhibitors of the GTPase KRASG12C in cancer: a patent review (2019-2021)EXPERT OPINION ON THERAPEUTIC PATENTS, 2022, 32 (05) : 475 - 505Xu, Qifu论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R ChinaZhang, Guozhen论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R ChinaLiu, Qian论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R ChinaLi, Shunda论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R ChinaZhang, Yingjie论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China Shandong Univ, Cheeloo Coll Med, Key Lab Chem Biol, Dept Med Chem,Sch Pharmaceut Sci,Minist Educ, 44 West Wenhua Rd, Jinan 250012, Peoples R China
- [46] SOS1 Inhibition Enhances the Efficacy of KRASG12C Inhibitors and Delays Resistance in Lung AdenocarcinomaCANCER RESEARCH, 2025, 85 (01) : 118 - 133Daley, Brianna R.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, USU Phys Scientist Training Program, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USASealover, Nancy E.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAFinniff, Bridget A.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAHughes, Jacob M.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USASheffels, Erin论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAGerlach, Daniel论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV GmbH & Co KG, Vienna, Austria Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAHofmann, Marco H.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV GmbH & Co KG, Vienna, Austria Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAKostyrko, Kaja论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim RCV GmbH & Co KG, Vienna, Austria Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USALamorte, Joseph P.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, USU Phys Scientist Training Program, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Anat Physiol & Genet, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USALinke, Amanda J.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USABeckley, Zaria论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAFrank, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: Henry M Jackson Fdn Advancement Mil Med, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Ctr Mil Precis Hlth, Student Bioinformat Initiat, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USALewis, Robert E.论文数: 0 引用数: 0 h-index: 0机构: Univ Nebraska Med Ctr, Eppley Inst Res Canc & Allied Dis, Omaha, NE USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAWilkerson, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Anat Physiol & Genet, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USADalgard, Clifton L.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Anat Physiol & Genet, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Amer Genome Ctr, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USAKortum, Robert L.论文数: 0 引用数: 0 h-index: 0机构: Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA Uniformed Serv Univ Hlth Sci, Dept Pharmacol & Mol Therapeut, Bethesda, MD USA
- [47] A next-generation KRASG12C inhibitor ABSK071 demonstrated broad synergy with other therapeutic agents in KRASG12C mutated cancer modelsCANCER RESEARCH, 2023, 83 (08)Ying, Haiyan论文数: 0 引用数: 0 h-index: 0Guo, Fushen论文数: 0 引用数: 0 h-index: 0Peng, Juan论文数: 0 引用数: 0 h-index: 0Wang, Jie论文数: 0 引用数: 0 h-index: 0Zhang, Jie论文数: 0 引用数: 0 h-index: 0Liu, Manqi论文数: 0 引用数: 0 h-index: 0Zhu, Zhixuan论文数: 0 引用数: 0 h-index: 0Chen, Zhui论文数: 0 引用数: 0 h-index: 0
- [48] Design, synthesis and bioactivity evaluation of novel quinazoline based KRASG12C inhibitorsNEW JOURNAL OF CHEMISTRY, 2022, 46 (10) : 4827 - 4836Liu, Qingxu论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R ChinaLi, Yan论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China Minist Hlth, Key Lab Biotech Drugs, Jinan 250117, Peoples R China Key Lab Rare & Uncommon Dis Shandong Prov, Jinan 250117, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R ChinaZhi, Ying论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China Minist Hlth, Key Lab Biotech Drugs, Jinan 250117, Peoples R China Key Lab Rare & Uncommon Dis Shandong Prov, Jinan 250117, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R ChinaLiu, Bo论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China Minist Hlth, Key Lab Biotech Drugs, Jinan 250117, Peoples R China Key Lab Rare & Uncommon Dis Shandong Prov, Jinan 250117, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R ChinaSun, Jingyong论文数: 0 引用数: 0 h-index: 0机构: Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China Minist Hlth, Key Lab Biotech Drugs, Jinan 250117, Peoples R China Key Lab Rare & Uncommon Dis Shandong Prov, Jinan 250117, Peoples R China Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250117, Peoples R China
- [49] Modeling receptor flexibility in the structure-based design of KRASG12C inhibitorsJournal of Computer-Aided Molecular Design, 2022, 36 : 591 - 604Kai Zhu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular EngineeringCui Li论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular EngineeringKingsley Y. Wu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular EngineeringChristopher Mohr论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular EngineeringXun Li论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular EngineeringBrian Lanman论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc.,Department of Molecular Engineering
- [50] The gRAss Is Greener: Potential new Therapies in Lung cancer with Acquired Resistance to KRAsG12c InhibitorsCANCER DISCOVERY, 2021, 11 (08) : 1874 - 1876Pinnelli, Marika论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Oncol, Turin, Italy Candiolo Canc Inst FPO IRCCS, Turin, Italy Univ Torino, Dept Oncol, Turin, ItalyTrusolino, Livio论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Oncol, Turin, Italy Candiolo Canc Inst FPO IRCCS, Turin, Italy Univ Torino, Dept Oncol, Turin, Italy