QUANTITATIVE PET-SCAN STUDIES ON HUMAN DOPAMINE-D2 RECEPTORS USING C-11 RACLOPRIDE, A SUBSTITUTED BENZAMIDE

被引:0
|
作者
FARDE, L
EHRIN, E
HALL, H
SEDVALL, G
机构
[1] KAROLINSKA INST,DEPT PSYCHIAT & PSYCHOL,S-10401 STOCKHOLM 60,SWEDEN
[2] ASTRA LAKEMEDEL AB,S-15185 SODERTALJE,SWEDEN
[3] KAROLINSKA PHARM,STOCKHOLM,SWEDEN
关键词
D O I
暂无
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:4 / 4
页数:1
相关论文
共 50 条
  • [41] LIGAND METABOLITES IN PLASMA DURING PET-STUDIES WITH THE C-11 LABELED DOPAMINE ANTAGONISTS, RACLOPRIDE, SCH 23390 AND N-METHYLSPIROPERIDOL
    SWAHN, CG
    FARDE, L
    HALLDIN, C
    SEDVALL, G
    HUMAN PSYCHOPHARMACOLOGY-CLINICAL AND EXPERIMENTAL, 1992, 7 (02) : 97 - 103
  • [42] Measurement of density and affinity for dopamine D2 receptors by a single positron emission tomography scan with multiple injections of [11C]raclopride
    Ikoma, Yoko
    Watabe, Hiroshi
    Hayashi, Takuya
    Miyake, Yoshinori
    Teramoto, Noboru
    Minato, Kotaro
    Iida, Hidehiro
    JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 2010, 30 (03): : 663 - 673
  • [43] Measurement of dopamine D2 receptors in living human brain using [11C] raclopride with ultra-high specific radioactivity
    Fujimura, Yota
    Ito, Hiroshi
    Takahashi, Hidehiko
    Yasuno, Fumihiko
    Ikoma, Yoko
    Zhang, Ming-Rong
    Nanko, Shinichiro
    Suzuki, Kazutoshi
    Suhara, Tetsuya
    NUCLEAR MEDICINE AND BIOLOGY, 2010, 37 (07) : 831 - 835
  • [44] Sleep deprivation decreases binding of [11C]raclopride to dopamine D2/D3 receptors in the human brain
    Volkow, Nora D.
    Wang, Gene-Jack
    Telang, Frank
    Fowler, Joanna S.
    Logan, Jean
    Wong, Christopher
    Ma, Jim
    Pradhan, Kith
    Tomasi, Dardo
    Thanos, Peter K.
    Ferre, Sergi
    Jayne, Millard
    JOURNAL OF NEUROSCIENCE, 2008, 28 (34): : 8454 - 8461
  • [45] C-11 AND I-125 IODOBENZAMIDE - A NEW LIGAND FOR PET AND SPECT IMAGING OF D2 DOPAMINE-RECEPTORS
    WONG, DF
    WILSON, AA
    DANNALS, RF
    RAVERT, HT
    GUNGON, R
    VILLEMAGNE, V
    LINKS, J
    WAGNER, HN
    JOURNAL OF NUCLEAR MEDICINE, 1987, 28 (06) : 1076 - 1076
  • [46] Effects of fluoxetine on dopamine D2 receptors in the human brain:: a positron emission tomography study with [11C]raclopride
    Penttilä, J
    Kajander, J
    Aalto, S
    Hirvonen, J
    Någren, K
    Ilonen, T
    Syvälahti, E
    Hietala, J
    INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY, 2004, 7 (04): : 431 - 439
  • [47] PREPARATION OF C-11-LABELLED RACLOPRIDE, A NEW POTENT DOPAMINE RECEPTOR ANTAGONIST - PRELIMINARY PET STUDIES OF CEREBRAL DOPAMINE-RECEPTORS IN THE MONKEY
    EHRIN, E
    FARDE, L
    DEPAULIS, T
    ERIKSSON, L
    GREITZ, T
    JOHNSTROM, P
    LITTON, JE
    NILSSON, JLG
    SEDVALL, G
    STONEELANDER, S
    OGREN, SO
    INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES, 1985, 36 (04): : 269 - &
  • [48] [C-11] NNC-112, A SELECTIVE PET RADIOLIGAND FOR EXAMINATION OF EXTRASTRIATAL DOPAMINE D1 RECEPTORS
    HALLDIN, C
    FOGED, C
    KARLSSON, P
    SWAHN, CG
    ANDERSON, PH
    FARDE, L
    JOURNAL OF NUCLEAR MEDICINE, 1994, 35 (05) : P122 - P122
  • [49] SYNTHESIS OF [METHOXY-H-3]- AND [METHOXY-C-11]- LABELED RACLOPRIDE - SPECIFIC DOPAMINE-D2 RECEPTOR LIGANDS
    EHRIN, E
    GAWELL, L
    HOGBERG, T
    DEPAULIS, T
    STROM, P
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1987, 24 (08): : 931 - 940
  • [50] Chronic subthalamic nucleus stimulation and striatal D2 dopamine receptors in Parkinson's disease -: A [11C]-raclopride PET study
    Thobois, S
    Fraix, V
    Savasta, M
    Costes, N
    Pollak, P
    Mertens, P
    Koudsie, A
    Le Bars, D
    Benabid, AL
    Broussolle, E
    JOURNAL OF NEUROLOGY, 2003, 250 (10) : 1219 - 1223