PHASE-TRANSFER MEDIATED SERINE O-ALKYLATION

被引：0
|
作者：
PALMER, MJ
DANILEWICZ, JC
VUONG, H
机构：
来源：
SYNLETT | 1994年 / 03期
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D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
N-Trityl-L-serine carboxylic esters are smoothly 0-alkylated without racemisation under phase transfer conditions. The process is most effective for activated electrophiles and offers significant improvement in terms of convenience, reproducibility and yield over literature procedures.
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页码：171 / 172
页数：2
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