SYNTHESIS AND BIOLOGICAL-ACTIVITY OF NOVEL NONSTEROIDAL PROGESTERONE-RECEPTOR ANTAGONISTS

被引:5
|
作者
HAMANN, LG
FARMER, LJ
JOHNSON, MG
GOLDMAN, ME
MAIS, DE
DAVTIAN, A
BENDER, SL
JONES, TK
机构
[1] Ligand Pharmaceuticals Inc., San Diego, California, 92121
来源
关键词
D O I
10.1111/j.1749-6632.1995.tb31398.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:383 / 387
页数:5
相关论文
共 50 条
  • [21] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF NOVEL INDOLYLIMIDAZOLINONES
    TRIVEDI, B
    SHAH, VH
    JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 1993, 70 (07) : 645 - 646
  • [22] Synthesis and biological activity of a novel, highly potent progesterone receptor antagonist
    Fuhrmann, U
    Hess-Stumpp, H
    Cleve, A
    Neef, G
    Schwede, W
    Hoffmann, J
    Fritzemeier, KH
    Chwalisz, K
    JOURNAL OF MEDICINAL CHEMISTRY, 2000, 43 (26) : 5010 - 5016
  • [23] THE PROGESTERONE-RECEPTOR - BIOLOGICAL EFFECTS OF PROGESTINS AND ANTIPROGESTINS
    SAVOURET, JF
    CHAUCHEREAU, A
    MISRAHI, M
    LESCOP, P
    MANTEL, A
    BAILLY, A
    MILGROM, E
    HUMAN REPRODUCTION, 1994, 9 : 7 - 11
  • [24] Synthesis and biological evaluation of cyclopentaquinoline derivatives as nonsteroidal glucocorticoid receptor antagonists
    Eda, Masahiro
    Kuroda, Tomoko
    Kaneko, Satoshi
    Aoki, Yoshiyuki
    Chieko, Okumura
    Ohbora, Tomoko
    Sakaue, Masaki
    Koyama, Natsumi
    Aritomo, Keiichi
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251
  • [25] Synthesis and Biological Evaluation of Cyclopentaquinoline Derivatives as Nonsteroidal Glucocorticoid Receptor Antagonists
    Eda, Masahiro
    Kuroda, Tomoko
    Kaneko, Satoshi
    Aoki, Yoshiyuki
    Yamashita, Masami
    Okumura, Chieko
    Ikeda, Yoshitaka
    Ohbora, Tomoko
    Sakaue, Masaki
    Koyama, Natsumi
    Aritomo, Keiichi
    JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (12) : 4918 - 4926
  • [26] MOLECULAR INTERACTION OF NONSTEROIDAL COMPOUNDS WITH UTERINE PROGESTERONE-RECEPTOR .1.
    AGNIHOTRI, A
    NEELIMA
    NIWAS, S
    BHAT, BK
    KUMAR, S
    SETH, M
    BHADURI, AP
    SRIVASTAVA, AK
    KAMBOJ, VP
    EXPERIMENTAL AND CLINICAL ENDOCRINOLOGY, 1986, 88 (02): : 185 - 192
  • [27] PROSTAGLANDINS AND PROGESTERONE-RECEPTOR ANTAGONISTS IN HUMAN-FERTILITY REGULATION
    HEALY, DL
    AUSTRALIAN & NEW ZEALAND JOURNAL OF OBSTETRICS & GYNAECOLOGY, 1994, 34 (03): : 357 - 360
  • [28] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A NOVEL ANALOG OF NITROFURANTOIN
    WHITE, RL
    BURROUS, SE
    SCHWAN, TJ
    JOURNAL OF PHARMACEUTICAL SCIENCES, 1977, 66 (02) : 277 - 278
  • [29] Novel mechanisms of progesterone antagonists and progesterone receptor
    Edwards, DP
    Leonhardt, SA
    Gass-Handel, E
    JOURNAL OF THE SOCIETY FOR GYNECOLOGIC INVESTIGATION, 2000, 7 (01) : S22 - S24
  • [30] Novel Mechanisms of Progesterone Antagonists and Progesterone Receptor
    Dean P. Edwards
    Susan A. Leonhardt
    Elizabeth Gass-Handel
    The Journal of the Society for Gynecologic Investigation: JSGI, 2000, 7 : S22 - S24