NONADRENERGIC [H-3] IDAZOXAN BINDING-SITES ARE PHYSICALLY DISTINCT FROM ALPHA-2-ADRENERGIC RECEPTORS

被引:0
|
作者
MICHEL, MC
REGAN, JW
GERHARDT, MA
NEUBIG, RR
INSEL, PA
MOTULSKY, HJ
机构
[1] UNIV CALIF SAN DIEGO,DEPT PHARMACOL,LA JOLLA,CA 92093
[2] DUKE UNIV,HOWARD HUGHES MED INST,DEPT MED,DURHAM,NC 27706
[3] UNIV MICHIGAN,SCH MED,DEPT PHARMACOL & MED,DIV HYPERTENS,ANN ARBOR,MI 48104
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:65 / 68
页数:4
相关论文
共 50 条
  • [41] INCREASED ALPHA-2-ADRENERGIC BINDING-SITES AND ANTILIPOLYTIC EFFECT IN ADIPOCYTES FROM GENETICALLY-OBESE RATS
    CARPENE, C
    REBOURCET, MC
    GUICHARD, C
    LAFONTAN, M
    LAVAU, M
    [J]. JOURNAL OF LIPID RESEARCH, 1990, 31 (05) : 811 - 819
  • [42] The novel alpha(2)-adrenoceptor agonist [H-3]mivazerol binds to non-adrenergic binding sites in human striatum membranes that are distinct from imidazoline receptors
    Flamez, A
    Gillard, M
    DeBacker, JP
    Vauquelin, G
    Noyer, M
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1997, 31 (01) : 125 - 129
  • [43] 3 DISTINCT BINDING-SITES FOR [H-3] PRAZOSIN IN THE RAT CEREBRAL-CORTEX
    OSHITA, M
    KIGOSHI, S
    MURAMATSU, I
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1991, 104 (04) : 961 - 965
  • [44] DISCRIMINATION BETWEEN ALPHA-2-ADRENOCEPTORS AND [H-3] IDAZOXAN-LABELED NONADRENERGIC SITES IN RABBIT WHITE FAT-CELLS
    LANGIN, D
    PARIS, H
    DAUZATS, M
    LAFONTAN, M
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION, 1990, 188 (4-5): : 261 - 272
  • [45] CHARACTERIZATION OF BINDING-SITES FOR [H-3] SPIROPERIDOL
    LUEDTKE, RR
    MOLINOFF, PB
    [J]. BIOCHEMICAL PHARMACOLOGY, 1987, 36 (19) : 3255 - 3264
  • [46] IDENTIFICATION AND CHARACTERIZATION OF ALPHA-2-ADRENERGIC RECEPTORS IN HUMAN MYOMETRIUM BY [RAUWOLSCINE-H-3 BINDING
    BOTTARI, SP
    VOKAER, A
    KAIVEZ, E
    LESCRAINIER, JP
    VAUQUELIN, G
    [J]. AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY, 1983, 146 (06) : 639 - 643
  • [47] IDENTIFICATION OF ALPHA-2 ADRENERGIC-RECEPTORS IN HUMAN FRONTAL-CORTEX MEMBRANES BY BINDING OF [H-3] RX-821002, THE 2-METHOXY ANALOG OF [H-3] IDAZOXAN
    VAUQUELIN, G
    DEVOS, H
    DEBACKER, JP
    EBINGER, G
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1990, 17 (04) : 537 - 546
  • [48] ALPHA-2-ADRENERGIC RECEPTORS IN PLATELET MEMBRANES OF DEPRESSED-PATIENTS - INCREASED AFFINITY FOR H-3 YOHIMBINE
    WOLFE, N
    COHEN, BM
    GELENBERG, AJ
    [J]. PSYCHIATRY RESEARCH, 1987, 20 (02) : 107 - 116
  • [49] SOLUBILIZED RECEPTORS FOR [H-3]DOPAMINE (D3 BINDING-SITES) FROM CANINE BRAIN
    DAVIS, A
    MADRAS, BK
    SEEMAN, P
    [J]. BIOCHEMICAL PHARMACOLOGY, 1982, 31 (07) : 1183 - 1187
  • [50] AUTORADIOGRAPHIC LOCALIZATION OF [H-3] ZOLPIDEM BINDING-SITES IN THE RAT CNS - COMPARISON WITH THE DISTRIBUTION OF [H-3] FLUNITRAZEPAM BINDING-SITES
    NIDDAM, R
    DUBOIS, A
    SCATTON, B
    ARBILLA, S
    LANGER, SZ
    [J]. JOURNAL OF NEUROCHEMISTRY, 1987, 49 (03) : 890 - 899