NONADRENERGIC [H-3] IDAZOXAN BINDING-SITES ARE PHYSICALLY DISTINCT FROM ALPHA-2-ADRENERGIC RECEPTORS

被引:0
|
作者
MICHEL, MC
REGAN, JW
GERHARDT, MA
NEUBIG, RR
INSEL, PA
MOTULSKY, HJ
机构
[1] UNIV CALIF SAN DIEGO,DEPT PHARMACOL,LA JOLLA,CA 92093
[2] DUKE UNIV,HOWARD HUGHES MED INST,DEPT MED,DURHAM,NC 27706
[3] UNIV MICHIGAN,SCH MED,DEPT PHARMACOL & MED,DIV HYPERTENS,ANN ARBOR,MI 48104
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:65 / 68
页数:4
相关论文
共 50 条
  • [1] [H-3] IDAZOXAN AND [H-3] RAUWOLSCINE BINDING OF CLONED HUMAN ALPHA-2-ADRENERGIC RECEPTORS
    MICHEL, MC
    REGAN, JW
    MOTULSKY, HJ
    INSEL, PA
    [J]. CLINICAL RESEARCH, 1989, 37 (02): : A527 - A527
  • [2] FURTHER PHARMACOLOGICAL CHARACTERIZATION OF [H-3] IDAZOXAN BINDING-SITES IN RAT-BRAIN - EVIDENCE FOR PREDOMINANT LABELING OF ALPHA-2-ADRENERGIC RECEPTORS
    RAYMON, HK
    SMITH, TD
    LESLIE, FM
    [J]. BRAIN RESEARCH, 1992, 582 (02) : 261 - 267
  • [3] NONADRENERGIC BINDING-SITES FOR THE ALPHA-2-ANTAGONIST [H-3] IDAZOXAN IN RABBIT URETHRAL SMOOTH-MUSCLE
    YABLONSKY, F
    LACOLLE, JY
    DAUSSE, JP
    [J]. JOURNAL OF RECEPTOR RESEARCH, 1991, 11 (1-4): : 153 - 162
  • [4] [H-3] IDAZOXAN AND SOME OTHER ALPHA-2-ADRENERGIC DRUGS ALSO BIND WITH HIGH-AFFINITY TO A NONADRENERGIC SITE
    MICHEL, MC
    BRODDE, OE
    SCHNEPEL, B
    BEHRENDT, J
    TSCHADA, R
    MOTULSKY, HJ
    INSEL, PA
    [J]. MOLECULAR PHARMACOLOGY, 1989, 35 (03) : 324 - 330
  • [5] BINDING OF [H-3] YOHIMBINE TO ALPHA-2-ADRENERGIC RECEPTORS IN RAT-LIVER
    ELREFAI, MF
    EXTON, JH
    [J]. FEDERATION PROCEEDINGS, 1981, 40 (03) : 245 - 245
  • [6] IMIDAZOLINE RECEPTORS, NONADRENERGIC IDAZOXAN BINDING-SITES AND ALPHA(2)-ADRENOCEPTORS IN THE HUMAN CENTRAL-NERVOUS-SYSTEM
    DEVOS, H
    BRICCA, G
    DEKEYSER, J
    DEBACKER, JP
    BOUSQUET, P
    VAUQUELIN, G
    [J]. NEUROSCIENCE, 1994, 59 (03) : 589 - 598
  • [7] ALPHA-2A ADRENOCEPTORS AND NONADRENERGIC IDAZOXAN BINDING-SITES IN CALF BRAIN AND RETINA ARE DISTINCT FROM THOSE IN HUMAN BRAIN
    VANLIEFDE, I
    VAUQUELIN, G
    DEKEYSER, J
    DEBACKER, JP
    DEVOS, H
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1993, 22 (05) : 501 - 509
  • [8] CHARACTERIZATION OF IMIDAZOLINE BINDING-SITES DISTINCT FROM ALPHA-2-ADRENERGIC RECEPTORS IN THE RABBIT IRIS-CILIARY BODY (ICB)
    LATOUR, E
    CALMETTE, C
    COQUELET, C
    [J]. INVESTIGATIVE OPHTHALMOLOGY & VISUAL SCIENCE, 1994, 35 (04) : 1889 - 1889
  • [9] DIFFERENCES IN THE REGULATION OF [H-3] IDAZOXAN AND [H-3] YOHIMBINE BINDING-SITES IN THE RABBIT
    YAKUBU, MA
    DEIGHTON, NM
    HAMILTON, CA
    REID, JL
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1990, 176 (03) : 305 - 311
  • [10] EVIDENCE THAT DRUG-BINDING TO NONADRENERGIC [H-3] IDAZOXAN BINDING-SITES (I-RECEPTORS) OCCURS TO INTERACTING OR INTERCONVERTIBLE AFFINITY FORMS OF THE RECEPTOR
    WIKBERG, JES
    UHLEN, S
    CHHAJLANI, V
    [J]. PHARMACOLOGY & TOXICOLOGY, 1992, 70 (03): : 208 - 219