ANTI-TUMOR AGENTS - DIAZOMETHYL KETONE AND CHLOROMETHYL KETONE ANALOGS PREPARED FROM N-TOSYL AMINO-ACIDS

被引：11
|
作者：
SAJADI, Z
KASHANI, M
LOEFFLER, LJ
HALL, IH
机构：
[1] UNIV N CAROLINA,SCH PHARM,DIV MED CHEM,CHAPEL HILL,NC 27514
[2] FERDOWSI UNIV,SCH PHARM,DIV MED CHEM,MESHHAD,IRAN
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1980年 / 23卷 / 03期
关键词：
D O I：
10.1021/jm00177a012
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：275 / 278
页数：4
相关论文
共 43 条
  • [11] IRREVERSIBLE INACTIVATION OF TRYPSIN BY CHLOROMETHYL KETONE DERIVED FROM N ALPHA-TOSYL-L-LYSINE
    MARESGUIA, M
    SHAW, E
    FEDERATION PROCEEDINGS, 1963, 22 (02) : 528 - &
  • [12] N-BENZOYL DERIVATIVES OF AMINO-ACIDS AND AMINO-ACID ANALOGS AS GROWTH-INHIBITORS IN MICROBIAL ANTI-TUMOR SCREEN
    OTANI, TT
    BRILEY, MR
    JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (11) : 1366 - 1369
  • [13] SYNTHESIS AND EVALUATION OF ANTI-TUMOR ACTIVITY OF NITROSOUREAS DERIVED FROM AMINO-ACIDS .2. FREE AMINO-ACIDS
    MONTERO, JL
    LEYDET, A
    MESSIEZMUNOZ, A
    DEWYNTER, G
    IMBACH, JL
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1984, 19 (06) : 512 - 518
  • [14] Asymmetric synthesis of N-tosyl amino acids from N-sulfinyl α-amino-1,3-dithioketals
    Davis, Franklin A.
    Ramachandar, Tokala
    Chai, Jing
    Qiu, Hiu
    ARKIVOC, 2010, : 17 - 26
  • [15] AMINO-ACIDS AND PEPTIDES .36. SYNTHESIS OF ENKEPHALIN CHLOROMETHYL KETONE AND EVALUATION OF ITS INHIBITORY ACTIVITY AGAINST ENDOPEPTIDASE 22.19
    TAGUCHI, H
    NISHIYAMA, Y
    CAMARGO, ACM
    OKADA, Y
    CHEMICAL & PHARMACEUTICAL BULLETIN, 1993, 41 (11) : 2038 - 2039
  • [16] STUDIES ON ACTIVE SITE OF CLOSTRIPAIN - SPECIFIC INACTIVATION BY CHLOROMETHYL KETONE DERIVED FROM ALPHA-N-TOSYL-L-LYSINE
    PORTER, WH
    CUNNINGH.LW
    MITCHELL, WM
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1971, 246 (24) : 7675 - +
  • [17] REMOVAL OF N-TOSYL AND N-BENZYLOXYCARBONYL PROTECTIVE GROUPS FROM AMINO-ACIDS BY ELECTROCHEMICAL REDUCTION IN DIMETHYLFORMAMIDE - STUDY OF AMINO-ACID ANIONS PROTONATION IN NON-AQUEOUS SOLUTION
    MAIRANOVSKY, VG
    LOGINOVA, NF
    BIOORGANICHESKAYA KHIMIYA, 1976, 2 (11): : 1497 - 1503
  • [18] ANTI-TUMOR EFFECT OF N-ALPHA-BENZYLOXYCARBONYL-N,N-BIS-(2-HALOGENETHYL)-HYDRAZIDE DERIVATIVES OF AMINO-ACIDS
    KARAIVANOVA, MH
    ZAKHARIEV, SG
    GOLOVINSKY, EV
    NEOPLASMA, 1980, 27 (02) : 137 - 142
  • [19] Synthesis and anti-tumor evaluation of novel 25-hydroxyprotopanaxadiol analogs incorporating natural amino acids
    Wang, Peng
    Bi, Xiu-Li
    Xu, Jing
    Yuan, Hao-Nan
    Piao, Hu-Ri
    Zhao, Yu-Qing
    STEROIDS, 2013, 78 (02) : 203 - 209
  • [20] Amino acids and peptides .48. Studies on the structure of an unexpected reaction product from dipeptidyl chloromethyl ketone during acid hydrolysis
    Yokoi, T
    Taguchi, H
    Nishiyama, Y
    Igarashi, K
    Kasuya, F
    Okada, Y
    JOURNAL OF CHEMICAL RESEARCH, 1997, (01) : 10 - 11
12345