BEHAVIOR OF 2-(BETA-SUBSTITUTED-ALPHA-BENZOYLAMINO)-(4H)-3,1-BENZOXAZIN-4-ONE TOWARDS SOME NUCLEOPHILES

被引：0
|
作者：
SOLIMAN, FMA
ESLAM, I
SOUKA, L
DAWOOD, N
机构：
来源：
JOURNAL OF THE CHEMICAL SOCIETY OF PAKISTAN | 1993年 / 15卷 / 02期
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中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Active methylene compounds react with 2-(alpha-benzoyl-amino-beta-p-chlorophenyl) vinyl (4H)-3,1-benzoxazin-4-one (1) to give the keto esters (2,3). Aromatic hydrocarbons react with (1) under Friedel-Crafts conditions to give the corresponding ketones (6 and 7). The reaction of (1) with phosphorus pentasulphide yields the corresponding thione (8). Reaction of (1) with sodium azide, Grignard reagents, and Diels-Alder has been described.
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页码：149 / 153
页数：5
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