AGONIST INTERACTIONS WITH THE ALPHA-ADRENERGIC RECEPTOR OF HUMAN-PLATELETS - HIGH-AFFINITY AGONIST BINDING REFLECTS THE EFFICIENCY OF MEMBRANE TRANSDUCTION

被引:0
|
作者
HOFFMAN, BB
MICHEL, T
LEFKOWITZ, RJ
机构
[1] DUKE UNIV,MED CTR,DEPT MED,DURHAM,NC 27710
[2] DUKE UNIV,MED CTR,DEPT BIOCHEM,DURHAM,NC 27710
来源
CLINICAL RESEARCH | 1981年 / 29卷 / 02期
关键词
D O I
暂无
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:A272 / A272
页数:1
相关论文
共 50 条
  • [31] The unique nature of thf serine interactions for alpha(1)-adrenergic receptor agonist binding and activation
    Hwa, J
    Perez, DM
    FASEB JOURNAL, 1996, 10 (03): : 2410 - 2410
  • [32] 3-Indoxyl sulfate is a high-affinity agonist of the human aryl hydrocarbon receptor
    Schroeder, Jennifer C.
    Murray, Iain A.
    Flaveny, Colin A.
    DiNatale, Brett C.
    Perdew, Gary H.
    DRUG METABOLISM REVIEWS, 2009, 41 : 170 - 170
  • [33] HIGH-AFFINITY BINDING OF [IMIPRAMINE-H-3 TO HUMAN-PLATELETS - COMPARISON WITH THE BINDING IN RAT-BRAIN
    BRILEY, M
    LANGER, SZ
    RAISMAN, R
    BRITISH JOURNAL OF PHARMACOLOGY, 1980, 69 (02) : P300 - P300
  • [34] DOPAMINE RECEPTOR-BINDING ON INTACT-CELLS - ABSENCE OF A HIGH-AFFINITY AGONIST-RECEPTOR BINDING STATE
    SIBLEY, DR
    MAHAN, LC
    CREESE, I
    MOLECULAR PHARMACOLOGY, 1983, 23 (02) : 295 - 302
  • [35] DELINEATION OF A REGION IN THE B2 BRADYKININ RECEPTOR THAT IS ESSENTIAL FOR HIGH-AFFINITY AGONIST BINDING
    NARDONE, J
    HOGAN, PG
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1994, 91 (10) : 4417 - 4421
  • [36] FORMATION OF THE HIGH-AFFINITY AGONIST STATE OF THE ALPHA-1-ADRENERGIC RECEPTOR AT COLD TEMPERATURES DOES NOT REQUIRE A G-PROTEIN
    LYNCH, CJ
    TAYLOR, SJ
    SMITH, JA
    EXTON, JH
    FEBS LETTERS, 1988, 229 (01) : 54 - 58
  • [37] PLASMA-CATECHOLAMINE MODULATION OF ALPHA-2 ADRENOCEPTOR AGONIST AFFINITY AND SENSITIVITY IN NORMOTENSIVE AND HYPERTENSIVE HUMAN-PLATELETS
    HOLLISTER, AS
    ONROT, J
    LONCE, S
    NADEAU, JHJ
    ROBERTSON, D
    JOURNAL OF CLINICAL INVESTIGATION, 1986, 77 (05): : 1416 - 1421
  • [38] Agonist-specific, high-affinity binding epitopes are contributed by an arginine in the N-terminus of the human oxytocin receptor
    Wesley, VJ
    Hawtin, SR
    Howard, HC
    Wheatley, M
    BIOCHEMISTRY, 2002, 41 (16) : 5086 - 5092
  • [39] HETEROGENEITY OF RADIOLIGAND BINDING TO ALPHA-ADRENERGIC RECEPTORS - ANALYSIS OF GUANINE-NUCLEOTIDE REGULATION OF AGONIST BINDING IN RELATION TO RECEPTOR SUBTYPES
    HOFFMAN, BB
    MULLIKINKILPATRICK, D
    LEFKOWITZ, RJ
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1980, 255 (10) : 4645 - 4652
  • [40] DEMONSTRATION OF SPECIFIC HIGH-AFFINITY BINDING-SITES FOR (H-3) IMIPRAMINE ON HUMAN-PLATELETS
    PAUL, SM
    REHAVI, M
    SKOLNICK, P
    GOODWIN, FK
    LIFE SCIENCES, 1980, 26 (12) : 953 - 959