AROMATASE INHIBITION BY 5-SUBSTITUTED PYRIMIDINES AND DIHYDROPYRIMIDINES

被引:24
|
作者
TAYLOR, HM [1 ]
JONES, CD [1 ]
DAVENPORT, JD [1 ]
HIRSCH, KS [1 ]
KRESS, TJ [1 ]
WEAVER, D [1 ]
机构
[1] ELI LILLY & CO,LILLY RES LAB,LILLY CORP CTR,INDIANAPOLIS,IN 46285
关键词
D O I
10.1021/jm00391a016
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1359 / 1365
页数:7
相关论文
共 50 条
  • [21] NICKEL CHELATES OF 5-SUBSTITUTED SALICYLALDEHYDE AND 5-SUBSTITUTED SALICYLALDOXIME LIGANDS
    KAPADIA, RN
    [J]. CURRENT SCIENCE, 1975, 44 (18): : 658 - 659
  • [22] Inhibition of Herpesvirus Replication by 5-Substituted 4′-Thiopyrimidine Nucleosides
    Prichard, Mark N.
    Quenelle, Debra C.
    Hartline, Caroll B.
    Harden, Emma A.
    Jefferson, Geraldine
    Frederick, Samuel L.
    Daily, Shannon L.
    Whitley, Richard J.
    Tiwari, Kamal N.
    Maddry, Joseph A.
    Secrist, John A., III
    Kern, Earl R.
    [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2009, 53 (12) : 5251 - 5258
  • [23] INHIBITION OF URICASE BY SUBSTITUTED PYRIMIDINES
    SEDOR, FA
    SANDER, EG
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 75 (02) : 406 - 413
  • [24] Synthesis and Topo I inhibition of 5-substituted camptothecins.
    Zhou, LM
    Zhou, YS
    Burgin, A
    Mo, XS
    Zembower, D
    Xie, YP
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2004, 228 : U929 - U929
  • [25] 5-SUBSTITUTED URACILS
    MULVEY, DM
    BABSON, RD
    ZAWOISKI, S
    RYDER, MA
    [J]. JOURNAL OF HETEROCYCLIC CHEMISTRY, 1973, 10 (01) : 79 - 83
  • [26] PYRIMIDINES .V. SOME HIGHER 5-SUBSTITUTED 2,4,6-TRICHLOROPYRIMIDINES
    GERSHON, H
    PARMEGIANI, R
    DASCOLI, R
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (01) : 113 - +
  • [27] CHEMOTHERAPEUTIC NITROHETEROCYCLES .24. 5-SUBSTITUTED 2-(5-NITRO-2-FURYL)PYRIMIDINES
    ALBRECHT, R
    SCHRODER, E
    [J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1975, 10 (06) : 595 - 598
  • [28] PHOTOREACTIONS OF DIAZINES .8. DI-PI-METHANE PHOTOREARRANGEMENT OF 4-SUBSTITUTED 1,4(OR 3,4)-DIHYDROPYRIMIDINES LEADING TO 5-SUBSTITUTED 1,2-DIHYDROPYRIMIDINES OR 2,3-DIHYDROPYRIMIDINES
    VANDERSTOEL, RE
    VANDERPLAS, HC
    [J]. JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1979, (05): : 1228 - 1232
  • [29] INHIBITION OF URACIL AND THYMINE DEGRADATION BY SOME 5-SUBSTITUTED URACIL ANALOGUES
    SEBESTA, K
    BAUEROVA, J
    SORMOVA, Z
    [J]. BIOCHIMICA ET BIOPHYSICA ACTA, 1961, 50 (02) : 393 - &
  • [30] Dihydrofolate reductase inhibition effect of 5-substituted pyrido[2,3-d] pyrimidines: Synthesis, antitumor activity and molecular modeling study
    Abdelaziz, Ola A.
    El Husseiny, Walaa M.
    Selim, Khalid B.
    Eisa, Hassan M.
    [J]. BIOORGANIC CHEMISTRY, 2019, 90