IMPROVED SYNTHESIS OF FLUOROALKYL AND FLUOROARYL SUBSTITUTED 2-AMINOPYRIMIDINES

被引：6
|
作者：
KUCEROVY, A
MATTNER, PG
HATHAWAY, JS
REPIC, O
机构：
[1] Chemical Research and Development, Sandoz Pharmaceuticals Corporation
来源：
SYNTHETIC COMMUNICATIONS | 1990年 / 20卷 / 06期
基金：
中国国家自然科学基金;
关键词：
D O I：
10.1080/00397919008052340
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Fluoroalkyl and fluoroaryl substituted 2-aminopyrimidines have been prepared in good yields by the cyclization of guanidine salts with fluorine substituted β-diketones in sodium isopropoxide/isopropanol at reflux. Copyright © 1990 by Taylor & Francis Group. All rights reserved.
引用
收藏
页码：913 / 917
页数：5
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