USE OF DICYCLOHEXYLCARBODIIMIDE/3-HYDROXY-4-OXO-3,4-DIHYDRO-CHINAZOLINE IN SYNTHESIS OF C-TERMINAL HEXAPEPTIDE AMIDE OF SUBSTANCE-P

被引：11
|
作者：
JAKUBKE, HD [1 ]
KLESSEN, C [1 ]
NEUBERT, K [1 ]
机构：
[1] MARTIN LUTHER UNIV,SEKT BIOWISSENSCH,DDR-402 HALLE,GER DEM REP
来源：
JOURNAL FUR PRAKTISCHE CHEMIE | 1977年 / 319卷 / 04期
关键词：
D O I：
10.1002/prac.19773190414
中图分类号：
O69 [应用化学];
学科分类号：
081704 ;
摘要：
引用
收藏
页码：640 / 646
页数：7
相关论文
共 18 条
  • [11] SYNTHESIS OF SUBSTANCE-P C-TERMINAL HEXAPEPTIDE ANALOGS AND THEIR BIOLOGICAL-ACTIVITY - ANALOGS WITH ANTAGONISTIC ACTIVITY WITHOUT CONTAINING D-AMINO ACIDS
    KARAGIANNIS, K
    MANOLOPOULOU, A
    POULOS, C
    STAVROPOULOS, G
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1994, 29 (09) : 667 - 673
  • [12] SYNTHESIS OF POTENT ANTAGONISTS OF SUBSTANCE-P BY MODIFYING THE METHIONYL AND GLUTAMINYL RESIDUES OF ITS C-TERMINAL HEXAPEPTIDE AND WITHOUT USING D-AMINO ACIDS
    MANOLOPOULOU, A
    KARAGIANNIS, K
    STAVROPOULOS, G
    POULOS, C
    JORDAN, CC
    HAGAN, RM
    INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH, 1993, 41 (04): : 411 - 414
  • [13] SYNTHESIS OF AN ANALOG OF THE SUBSTANCE-P C-TERMINAL HEXAPEPTIDE WITH MODIFICATION AT THE GLUTAMINYL AND METHIONINYL RESIDUES AND INCREASED ACTIVITY IN NK-2 RECEPTOR TYPE - STRUCTURE-ACTIVITY-RELATIONSHIPS
    MANOLOPOULOU, A
    POULOS, C
    TSEGENIDIS, T
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1992, 27 (09) : 949 - 954
  • [14] Synthesis of 3,4-dihydro-3-hydroxy-10-oxo-10H-[2,3-C]benzodipyrans with hydrogen peroxide catalyzed by PCWP oxidative cyclization of 4-allyl-3-hydroxycoumarins.
    Suraparaju, RR
    Krupadanam, GLD
    Srimannarayana, G
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U186 - U186
  • [15] 2-Acyl(aroyl)-1,1,3,3-tetracyanopropenides 7*. Synthesis of 4-amino-1-aryl-6-halo-1-hydroxy-3-oxo-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-7-carbonitriles
    Kayukov, Yakov S.
    Karpov, Sergey V.
    Grigor'ev, Arthur A.
    Nikiforova, Anastasiya L.
    Nasakin, Oleg E.
    Shchegravina, Ekaterina S.
    Kayukova, Olga V.
    Tafeenko, Victor A.
    CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2017, 53 (05) : 568 - 574
  • [16] Interaction of 3-p-toluoyl-1,2-dihydro-4H-pyrrolo-[2,1-c][1,4]benzoxazine-1,2,4-trione with benzylamine. Synthesis and crystal and molecular structure ofZ-3-(1-benzyl-2-hydroxy-4,5-dioxo-2-p-tolyltetrahydropyrrol-3-idene)-3,4-dihydro-2H-1,4-benzoxazin-2-one
    Z. G. Aliev
    A. N. Maslivets
    I. V. Mashevskaya
    Yu. S. Andreichikov
    L. O. Atovmyan
    Russian Chemical Bulletin, 1997, 46 : 546 - 549
  • [17] Interaction of 3-p-toluoyl-1,2-dihydro-4H-pyrrolo[2,1-c][1,4]benzoxazine-1,2,4-trione with benzylamine. Synthesis and crystal and molecular structure of Z-3-(1-benzyl-2-hydroxy-4,5-dioxo-2-p-tolyltetrahydropyrrol-3-idene)-3,4-dihydro-2H-1,4-benzoxazin-2-one
    Aliev, ZG
    Maslivets, AN
    Mashevskaya, IV
    Andreichikov, YS
    Atovmyan, LO
    RUSSIAN CHEMICAL BULLETIN, 1997, 46 (03) : 546 - 549
  • [18] Design and synthesis of highly potent benzodiazepine γ-secretase inhibitors:: Preparation of (2S,3R)-3-(3,4-difluorophenyl)-2-(4-fluorophenyl)-4-hydroxy-N-((3S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]- diazepin-3-yl)butyramide by use of an asymmetric Ireland-Claisen rearrangement
    Churcher, I
    Williams, S
    Kerrad, S
    Harrison, T
    Castro, JL
    Shearman, MS
    Lewis, HD
    Clarke, EE
    Wrigley, JDJ
    Beher, D
    Tang, YS
    Liu, WS
    JOURNAL OF MEDICINAL CHEMISTRY, 2003, 46 (12) : 2275 - 2278
12