2-STEP SYNTHESIS OF SUBSTITUTED INDOLO[1,2-A]-QUINOXALIN-6-ONES

被引：20
|
作者：
BEACH, MJ [1 ]
HOPE, R [1 ]
KLAUBERT, DH [1 ]
RUSSELL, RK [1 ]
机构：
[1] RW JOHNSON PHARMACEUT RES INST,RARITAN,NJ 08869
来源：
SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 14期
关键词：
D O I：
10.1080/00397919508015898
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reaction of indole-2-carboxylates with 2-fluoronitrobenzenes in 1-methyl-2-pyrrolidinone containing NaH affords the 1-(2-nitrophenyl)indole-2-carboxlyates 1. These compounds are reduced with iron in acetic acid to afford the indolo[1,2-a]quinoxalin-6(5H)-ones 2.
引用
收藏
页码：2165 / 2183
页数：19
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