Synthesis of pyrazino[1,2-a]indoles and indolo-[1,2-a]quinoxalines (microreview)

被引：11
|
作者：
Sokolova, Ekaterina A. [1 ]
Festa, Alexey A. [1 ]
机构：
[1] Peoples Friendship Univ Russia, 6 Miklukho Maklaya St, Moscow 117198, Russia
来源：
CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2016年 / 52卷 / 04期
关键词：
INTRAMOLECULAR CYCLIZATION; DERIVATIVES;
D O I：
10.1007/s10593-016-1866-y
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The review is dedicated to the methods of synthesis of pyrazino[1,2-a]indoles and indolo[1,2-a]-quinoxalines. The primary approach to the synthesis of these heterocyclic systems is the annulation of a pyrazine ring to a functionalized indole ring by means of condensation of carbonyl compounds, radical reactions catalyzed by transition metals, as well as hypervalent iodine compounds.
引用
收藏
页码：219 / 221
页数：3
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