SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 3-(4'-ARYL-2'-THIAZOLYL)-2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINES AND 2-(4'-ARYL-2'-THIAZOLYLAMINO)-4-OXO-4H-3,1-BENZOXAZINES FROM METHYL N-(4-ARYL-2-THIAZOLYL)DITHIOCARBAMATES

被引：0
|
作者：
KHAN, RH
RASTOGI, RC
机构：
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1993年 / 32卷 / 05期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reaction of methyl N-(4-aryl-2-thiazolyl)dithiocarbamates (2) with potassium anthranilate (1) in dimethylformamide below room temperature yields benzoxazines (6) whereas in refluxing dimethylformamide affords the isomeric tetrahydroquinazolines (5). The antifungal and antibacterial activities of these compounds have also been evaluated.
引用
收藏
页码：595 / 598
页数：4
相关论文
共 50 条
  • [41] ON THE ACIDITY OF 3-ARYL-4-OXO-2-THIOXO-1,2,3,4-TETRAHYDROQUINAZOLINONES
    RULKE, H
    MARTIN, E
    KOTTKE, K
    KUHMSTEDT, H
    PHARMAZIE, 1990, 45 (11): : 862 - 863
  • [42] PREPARATION DE QUELQUES ALCOYL-3 ARYL-2 OXO-4 DIHYDROBENZOTHIAZINES-1,3
    MOREAU, RC
    DELACOUX, E
    BULLETIN DE LA SOCIETE CHIMIQUE DE FRANCE, 1962, (03): : 502 - &
  • [43] HETEROCYCLES IN ORGANIC-SYNTHESIS .6. - A FACILE SYNTHESIS OF "1-(4-ARYL-2-THIAZOLYL)-2-PROPANONES
    SINGH, H
    AGGARWAL, SK
    MALHOTRA, N
    HETEROCYCLES, 1984, 22 (02) : 353 - 354
  • [44] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 3-(3'-CARBOXYPHENYLSULPHONAMIDO)-2-ARYL-5H-4-THIAZOLIDINONE
    JOSHI, SN
    SHAH, KD
    CHAUHAN, NA
    BAXI, AJ
    JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 1991, 68 (11) : 627 - 628
  • [45] Synthesis of N-[aryl(4-hydroxy-6-methyl-2-oxo-2H-pyran-3-yl)methyl] thioacetamide derivatives
    Zhiani, Rahele
    JOURNAL OF CHEMICAL RESEARCH, 2016, (01) : 26 - 28
  • [46] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF BIS-(2-ARYL-4-OXO-4H-CHROMEN-3-YL) SULFONES
    Ramesh, P.
    Jeyachandran, M.
    Durgashankar, R.
    INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2009, 18 (03) : 211 - 214
  • [47] 4-OXO-1,2,3,4-TETRAHYDROQUINAZOLINES .3. SYNTHESIS AND CHOLERETIC ACTIVITY OF QUINAZOLINE DERIVATIVES
    OKUMURA, K
    OINE, T
    OCHIAI, T
    TANI, J
    YAMADA, Y
    INOUE, I
    JOURNAL OF MEDICINAL CHEMISTRY, 1972, 15 (05) : 518 - &
  • [48] SYNTHESIS OF 2-ARYL + 2-ARYL-3-METHYL-DECAHYDRO-QUINOLIN-4-ONES
    BALIAH, V
    NATARAJAN, A
    INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1981, 20 (09): : 830 - 830
  • [49] Synthesis and antibacterial activity of tert-butyl [1-benzyl-2[(4-aryl-2-thiazolyl)hydrazono]ethyl]carbamate derivatives
    Turan-Zitouni, Gulhan
    Fehrentz, Jean-Alain
    Chevallet, Pierre
    Martinez, Jean
    Kaplancikli, Zafer Asim
    Ozdemir, Ahmet
    Arslanyolu, Muhittin
    Yildiz, Mehmet Taha
    ARCHIV DER PHARMAZIE, 2007, 340 (06) : 310 - 314
  • [50] Synthesis and evaluation of anticancer and antiviral activity of some 2-aryl-3(4-(2H-1-benzopyran-2-one-3-yl)-2-thiazolyl)-5-methyl-4-thiazolidinones
    Rao, VR
    Kumar, PV
    Reddy, VR
    Reddy, KM
    HETEROCYCLIC COMMUNICATIONS, 2005, 11 (3-4) : 273 - 284
12345