PYRIDAZINES .57. SYNTHESIS AND CYCLOCONDENSATION REACTIONS OF (2-AMINOPHENYL)-(4-PYRIDAZINYL)-KETONE, A NEW DIAZA ISOSTER OF 2-AMINOBENZOPHENONE

被引：6
|
作者：
HAIDER, N
HEINISCH, G
MOSHUBER, J
机构：
[1] Institute of Pharmaceutical Chemistry, University of Vienna, Vienna, A-1090
来源：
ARCHIV DER PHARMAZIE | 1992年 / 325卷 / 02期
关键词：
D O I：
10.1002/ardp.19923250212
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A convenient approach to the new 2-aminobenzophenone analogue 4 is reported. Condensation reactions of 4 with ortho esters or amide acetals, respectively, followed by intramolecular cyclisations were found to provide smooth access to (4-pyridazinyl)-substituted quinolines 10, 13a,b and the quinazoline derivative 15.
引用
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页码：119 / 122
页数：4
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