DIAZOCYCLOHEXADIENONES AS PHOTOAFFINITY LIGANDS - SYNTHESES OF TRIOXABICYCLOOCTANE PROBES FOR THE CONVULSANT BINDING-SITE OF THE GABAA RECEPTOR

被引：13
|
作者：
GOELDNER, MP
HAWKINSON, JE
CASIDA, JE
机构：
来源：
TETRAHEDRON LETTERS | 1989年 / 30卷 / 07期
关键词：
D O I：
10.1016/S0040-4039(01)80625-0
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
引用
收藏
页码：823 / 826
页数：4
相关论文
共 50 条
  • [1] Impact of membrane cholesterol on binding properties of benzodiazepine and convulsant site ligands to the GABAA receptor:: A discrete binding site?
    Bailey, BW
    Lewis, J
    Mitchell, DC
    BIOPHYSICAL JOURNAL, 2004, 86 (01) : 253A - 253A
  • [2] PHOTOAFFINITY LIGANDS FOR THE [H-3] TBOB BINDING-SITE OF THE GABA-A RECEPTOR
    HAWKINSON, JE
    GOELDNER, MP
    PALMER, CJ
    CASIDA, JE
    JOURNAL OF RECEPTOR RESEARCH, 1991, 11 (1-4): : 391 - 405
  • [3] PHOTOAFFINITY PROBES OF THE ALLYLIC PYROPHOSPHATE BINDING-SITE OF UNDECAPRENYL PYROPHOSPHATE SYNTHETASE
    ALLEN, CM
    BABA, T
    FEDERATION PROCEEDINGS, 1983, 42 (07) : 1910 - 1910
  • [4] Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands
    Richter L.
    De Graaf C.
    Sieghart W.
    Varagic Z.
    Mörzinger M.
    De Esch I.J.P.
    Ecker G.F.
    Ernst M.
    Nature Chemical Biology, 2012, 8 (5) : 455 - 464
  • [5] Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands
    Richter, Lars
    de Graaf, Chris
    Sieghart, Werner
    Varagic, Zdravko
    Moerzinger, Martina
    de Esch, Iwan J. P.
    Ecker, Gerhard F.
    Ernst, Margot
    NATURE CHEMICAL BIOLOGY, 2012, 8 (05) : 455 - 464
  • [6] Identification of the Functional Binding Site for the Convulsant Tetramethylenedisulfotetramine in the Pore of the α2β3γ2 GABAA Receptor
    Pressly, Brandon
    Lee, Ruth D.
    Barnych, Bogdan
    Hammock, Bruce D.
    Wulff, Heike
    MOLECULAR PHARMACOLOGY, 2021, 99 (01) : 78 - 91
  • [7] DESIGN OF A PHOTOAFFINITY LABEL FOR HORMONE BINDING-SITE OF NEUROPHYSIN
    KLAUSNER, YS
    MCCORMICK, WM
    CHAIKEN, IM
    INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH, 1978, 11 (01): : 82 - 90
  • [8] PHOTOAFFINITY-LABELING OF THE ACTIN NUCLEOTIDE BINDING-SITE
    HEGYI, G
    SZILAGYI, L
    JOURNAL OF MUSCLE RESEARCH AND CELL MOTILITY, 1984, 5 (02) : 193 - 193
  • [9] Photoaffinity labeling in target- and binding-site identification
    Smith, Ewan
    Collins, Ian
    FUTURE MEDICINAL CHEMISTRY, 2015, 7 (02) : 159 - 183
  • [10] PHOTOAFFINITY-LABELING OF THE NUCLEOTIDE BINDING-SITE OF ACTIN
    HEGYI, G
    SZILAGYI, L
    ELZINGA, M
    BIOCHEMISTRY, 1986, 25 (19) : 5793 - 5798
12345