SYNTHESIS OF POTENT ANTI-HIV AGENTS - ESTERS OF CASTANOSPERMINE

被引：40
|
作者：
LIU, PS [1 ]
HOEKSTRA, WJ [1 ]
KING, CHR [1 ]
机构：
[1] MERRELL DOW RES INST,INDIANAPOLIS,IN 46268
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 20期
关键词：
D O I：
10.1016/0040-4039(90)80159-J
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The syntheses of 6-0- and 7-0-acyl derivatives of the indolizidine alkaloid castanospermine, are described. These compounds are potent inhibitors of the human immunodeficiency virus (HIV) and are potential anti-AIDS agents. © 1990.
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页码：2829 / 2832
页数：4
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