CERTAIN STEROIDAL (3,4-C)-1',2',5'-OXADIAZOLES

被引：0
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作者：
YADAV, MR
JINDAL, DP
机构：
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1991年 / 30卷 / 05期
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O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Synthesis of some potential antiprogestational steroidal [3,4-c]-1',2',5'-oxadiazoles (1-4) is described. Testosterone acetate affords 7 involving a number of steps. 7 on Jones' oxidation followed by allylation gives 1. Similarly 2 and 3 have been obtained from their respective 17-oxo compounds. 17-alpha-Hydroxy derivative (4) has been prepared through two different routes starting from 16-alpha, 17-alpha-oxido compound 8.
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页码：473 / 476
页数：4
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