CATECHOL O-METHYLTRANSFERASE .2. IN-VITRO INHIBITION BY SUBSTITUTED 8-HYDROXYQUINOLINES

被引：37
|
作者：
BORCHARDT, RT [1 ]
机构：
[1] UNIV KANSAS, DEPT BIOCHEM, MCCOLLUM LABS, LAWRENCE, KS 66044 USA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1973年 / 16卷 / 04期
关键词：
D O I：
10.1021/jm00262a016
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：382 / 387
页数：6
相关论文
共 50 条
  • [1] Optimization of 8-Hydroxyquinolines as Inhibitors of Catechol O-Methyltransferase
    Buchler, Ingrid
    Akuma, Daniel
    Au, Vinh
    Carr, Gregory
    de Leon, Pablo
    DePasquale, Michael
    Ernst, Glen
    Huang, Yifang
    Kimos, Martha
    Kolobova, Anna
    Poslusney, Michael
    Wei, Huijun
    Swinnen, Dominique
    Montel, Florian
    Moureau, Florence
    Jigorel, Emilie
    Schulze, Monika-Sarah E. D.
    Wood, Martyn
    Barrow, James C.
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (21) : 9647 - 9665
  • [2] CATECHOL O-METHYLTRANSFERASE .8. STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION BY 8-HYDROXYQUINOLINES
    BORCHARDT, RT
    THAKKER, DR
    WARNER, VD
    MIRTH, DB
    SANE, JN
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1976, 19 (04) : 558 - 560
  • [3] A semiempirical study on inhibition of catechol O-methyltransferase by substituted catechols
    Ovaska, M
    Yliniemela, A
    [J]. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 1998, 12 (03) : 301 - 307
  • [4] A semiempirical study on inhibition of catechol O-methyltransferase by substituted catechols
    Martti Ovaska
    Ari Yliniemelä
    [J]. Journal of Computer-Aided Molecular Design, 1998, 12 : 301 - 307
  • [5] INHIBITION OF O-METHYLTRANSFERASE BY CATECHOL AND SENSITIZATION TO EPINEPHRINE
    BACQ, ZM
    GOSSELIN, L
    DRESSE, A
    RENSON, J
    [J]. SCIENCE, 1959, 130 (3373) : 453 - 454
  • [6] 8-HYDROXYQUINOLINES - IN-VITRO ANTIPLAQUE ACTIVITY AND PARTITION-COEFFICIENTS
    MIRTH, DB
    WARNER, VD
    PASTORE, MP
    [J]. JOURNAL OF DENTAL RESEARCH, 1973, 52 : 98 - &
  • [7] CATECHOL O-METHYLTRANSFERASE .1. KINETICS OF TROPOLONE INHIBITION
    BORCHARDT, RT
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (04) : 377 - 382
  • [8] AUGMENTATION OF PRESSOR RESPONSE TO GUANETHEDINE BY INHIBITION OF CATECHOL O-METHYLTRANSFERASE
    WYLIE, DW
    [J]. NATURE, 1961, 189 (476) : 490 - +
  • [9] The inhibition of catechol O-methyltransferase and monoamine oxidase by tetralone and indanone derivatives substituted with the nitrocatechol moiety
    de Beer, Andries D.
    Legoabe, Lesetja J.
    Petzer, Anel
    Petzer, Jacobus P.
    [J]. BIOORGANIC CHEMISTRY, 2021, 114
  • [10] ABSORPTION SPECTRA OF COPPER(2) AND NICKEL(2) COMPLEXES OF SUBSTITUTED 8-HYDROXYQUINOLINES
    MORPURGO, L
    WILLIAMS, RJP
    [J]. JOURNAL OF THE CHEMICAL SOCIETY A -INORGANIC PHYSICAL THEORETICAL, 1966, (01): : 73 - +
12345