A PYRIDAZINYL DERIVATIVE OF GAMMA-AMINOBUTYRIC-ACID (GABA), SR-95531, IS A POTENT ANTAGONIST OF CL- CHANNEL OPENING REGULATED BY GABA-A RECEPTORS

被引：30

|

作者：

MIENVILLE, JM

VICINI, S

机构：

来源：

NEUROPHARMACOLOGY | 1987年 / 26卷 / 7A期

关键词：

D O I：

10.1016/0028-3908(87)90242-5

中图分类号：

Q189 [神经科学];

学科分类号：

071006 ;

摘要：

引用

收藏

页码：779 / 783

页数：5

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[1] GAMMA-AMINOBUTYRIC-ACID GATING OF CL- CHANNELS IN RECOMBINANT GABA(A) RECEPTORS
DUCIC, I
CARUNCHO, HJ
ZHU, WJ
VICINI, S
COSTA, E
[J]. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1995, 272 (01): : 438 - 445
[2] QUANTITATIVE-EVALUATION OF THE PROPERTIES OF A PYRIDAZINYL GABA DERIVATIVE (SR-95531) AS A GABAA COMPETITIVE ANTAGONIST - AN ELECTROPHYSIOLOGICAL APPROACH
HAMANN, M
DESARMENIEN, M
DESAULLES, E
BADER, MF
FELTZ, P
[J]. BRAIN RESEARCH, 1988, 442 (02) : 287 - 296
[3] POTENTIATORS OF RESPONSES TO ACTIVATION OF GAMMA-AMINOBUTYRIC-ACID (GABA-A) RECEPTORS
SIMMONDS, MA
TURNER, JP
[J]. NEUROPHARMACOLOGY, 1987, 26 (7B) : 923 - 930
[4] INHIBITION OF LUTEINIZING-HORMONE SECRETION IN OVARIECTOMIZED EWES DURING THE BREEDING-SEASON BY GAMMA-AMINOBUTYRIC-ACID (GABA) IS MEDIATED BY GABA-A RECEPTORS, BUT NOT GABA-B RECEPTORS
SCOTT, CJ
CLARKE, IJ
[J]. ENDOCRINOLOGY, 1993, 132 (04) : 1789 - 1796
[5] MURINE RENAL MEDULLARY CL- CHANNELS ARE SIMILAR IN CDNA SEQUENCE TO A GAMMA-AMINOBUTYRIC-ACID (GABA)-ALPHA CL- CHANNEL IN THE CENTRAL-NERVOUS-SYSTEM (CNS)
MOLONY, D
BURGES, A
DUBOSE, T
MEHTA, P
[J]. FASEB JOURNAL, 1993, 7 (03): : A352 - A352
[6] CAN CL- IONS BE EXTRUDED FROM A GAMMA-AMINOBUTYRIC (GABA)-ACCEPTIVE NERVE-CELL VIA GABA-A RECEPTORS ON THE PLASMA-MEMBRANE CYTOPLASMIC SIDE
CUPELLO, A
PALM, A
RAPALLINO, MV
HYDEN, H
[J]. CELLULAR AND MOLECULAR NEUROBIOLOGY, 1991, 11 (03) : 333 - 346
[7] RENAL LOCALIZATION OF MESSENGER-RNA FOR A MURINE GAMMA-AMINOBUTYRIC-ACID (GABA)A ALPHA-1 CL- CHANNEL AND INCREASED EXPRESSION AFTER IN-VIVO PESTICIDE EXPOSURE
MOLONY, D
HAMILTON, R
HOLIAN, A
MEHTA, PS
[J]. JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, 1994, 5 (03): : 294 - 294
[8] CHARACTERIZATION OF BICUCULLINE BACLOFEN-INSENSITIVE GAMMA-AMINOBUTYRIC-ACID RECEPTORS EXPRESSED IN XENOPUS OOCYTES .1. EFFECTS OF CL- CHANNEL INHIBITORS
WOODWARD, RM
POLENZANI, L
MILEDI, R
[J]. MOLECULAR PHARMACOLOGY, 1992, 42 (01) : 165 - 173
[9] GAMMA-AMINOBUTYRIC-ACID (GABA)-MEDICATED AND BARBITURATE-MEDIATED CL-36(-) UPTAKE IN RAT-BRAIN SYNAPTONEUROSOMES - EVIDENCE FOR RAPID DESENSITIZATION OF THE GABA RECEPTOR-COUPLED CHLORIDE-ION CHANNEL
SCHWARTZ, RD
SUZDAK, PD
PAUL, SM
[J]. MOLECULAR PHARMACOLOGY, 1986, 30 (05) : 419 - 426
[10] GAMMA-AMINOBUTYRIC-ACID, THROUGH GABA-A RECEPTORS, INHIBITS THE POTASSIUM-STIMULATED RELEASE OF CALCITONIN GENE-RELATED PEPTIDE BUT NOT THAT OF SUBSTANCE-P-LIKE MATERIAL FROM RAT SPINAL-CORD SLICES
BOURGOIN, S
POHL, M
BENOLIEL, JJ
MAUBORGNE, A
COLLIN, E
HAMON, M
CESSELIN, F
[J]. BRAIN RESEARCH, 1992, 583 (1-2) : 344 - 348