BROP - A NEW REAGENT FOR COUPLING N-METHYLATED AMINO-ACIDS

被引：108
|
作者：
COSTE, J
DUFOUR, MN
PANTALONI, A
CASTRO, B
机构：
[1] Centre CNRS-INSERM de Pharmacologie Endocrinologie, 34094 Montpellier Cédex 2, Rue de la Cardonille
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 05期
关键词：
D O I：
10.1016/S0040-4039(00)94598-2
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
BroP (bromo tris(dimethylamino) phosphonium hexafluorophosphate) is a particularly suitable reagent for coupling N-methylated amino acids. It is stable and gives very high yields in short reaction times. Dipeptides are obtained without appreciable epimerization. © 1990.
引用
收藏
页码：669 / 672
页数：4
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