EFFECT OF DEUTERATION OF IMIPRAMINE ON ITS PHARMACOKINETIC PROPERTIES IN THE RAT

被引:13
|
作者
TAYLOR, IW
IOANNIDES, C
SACRA, P
TURNER, JC
PARKE, DV
机构
[1] UNIV SURREY,DEPT BIOCHEM,GUILDFORD GU2 5XH,SURREY,ENGLAND
[2] BIOREX LABS LTD,LONDON N1 2HB,ENGLAND
关键词
D O I
10.1016/0006-2952(83)90488-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:641 / 647
页数:7
相关论文
共 50 条
  • [1] BUCCAL ABSORPTION AND OTHER PROPERTIES OF PHARMACOKINETIC IMPORTANCE OF IMIPRAMINE AND ITS METABOLITES
    BICKEL, MH
    WEDER, HJ
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 1969, 21 (03) : 160 - &
  • [2] Effect of deuteration on the single dose pharmacokinetic properties and postoperative analgesic activity of methadone
    Wang, Xiao-ming
    Wang, Jigong
    Fokina, Valentina
    Patrikeeva, Svetlana
    Rytting, Erik
    Ahmed, Mahmoud S.
    La, Jun-Ho
    Nanovskaya, Tatiana
    DRUG METABOLISM AND PHARMACOKINETICS, 2022, 47
  • [3] MICRO-DETERMINATION OF GLYCERYL TRINITRATE IN BIOLOGICAL-FLUIDS - EFFECT OF DEUTERATION OF GLYCERYL TRINITRATE ON ITS PHARMACOKINETIC PROPERTIES
    TAYLOR, IW
    IOANNIDES, C
    TURNER, JC
    KOENIGSBERGER, RU
    PARKE, DV
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 1981, 33 (04) : 244 - 246
  • [4] MEASUREMENT AND PHARMACOKINETIC ANALYSIS OF IMIPRAMINE AND ITS METABOLITE BY BRAIN MICRODIALYSIS
    SATO, Y
    SHIBANOKI, S
    SUGAHARA, M
    ISHIKAWA, K
    BRITISH JOURNAL OF PHARMACOLOGY, 1994, 112 (02) : 625 - 629
  • [5] RELATIONSHIP BETWEEN REGIONAL DISTRIBUTION OF IMIPRAMINE AND ITS EFFECT ON LEARNED HELPLESSNESS IN THE RAT
    SHERMAN, AD
    ALLERS, GL
    NEUROPHARMACOLOGY, 1980, 19 (02) : 159 - 162
  • [6] CORRELATIVE CHANGES OF SEROTONIN AND CATECHOLAMINES WITH PHARMACOKINETIC ALTERATIONS OF IMIPRAMINE IN RAT-BRAIN
    SUGITA, S
    KOBAYASHI, A
    SUZUKI, S
    YOSHIDA, T
    NAKAZAWA, K
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1989, 165 (2-3) : 191 - 198
  • [7] The Effect of Deuteration and Homologation of the Lactam Ring of Nirmatrelvir on Its Biochemical Properties and Oxidative Metabolism
    Arutyunova, Elena
    Belovodskiy, Alexandr
    Chen, Pu
    Khan, Muhammad Bashir
    Joyce, Michael
    Saffran, Holly
    Lu, Jimmy
    Turner, Zoe
    Bai, Bing
    Lamer, Tess
    Young, Howard S.
    Vederas, John C.
    Tyrrell, D. Lorne
    Lemieux, M. Joanne
    Nieman, James A.
    ACS BIO & MED CHEM AU, 2023, 3 (06): : 528 - 541
  • [8] Effect of deuteration on the quadratic electrooptic properties of KDP
    Ledzion, R
    Bondarczuk, K
    Górski, P
    Kucharczyk, W
    CRYSTAL RESEARCH AND TECHNOLOGY, 1999, 34 (5-6) : 745 - 749
  • [9] EFFECT OF DEUTERATION ON ELECTROOPTIC PROPERTIES OF KDP CRYSTALS
    VLOKH, OG
    LUTSIVSH.LF
    OSTAPCHU.VP
    FIZIKA TVERDOGO TELA, 1974, 16 (01): : 271 - 273
  • [10] THE EFFECT OF IMIPRAMINE ON RAT DETRUSOR MUSCLE CONTRACTILITY
    OLUBADEWO, JO
    ARCHIVES INTERNATIONALES DE PHARMACODYNAMIE ET DE THERAPIE, 1980, 245 (01): : 84 - 94