MODULATION OF ANXIETY BY BETA-CARBOLINES AND OTHER BENZODIAZEPINE RECEPTOR LIGANDS - RELATIONSHIP OF PHARMACOLOGICAL TO BIOCHEMICAL MEASURES OF EFFICACY

被引:70
|
作者
STEPHENS, DN
SCHNEIDER, HH
KEHR, W
JENSEN, LH
PETERSEN, E
HONORE, T
机构
[1] SCHERING AG, RES LABS, D-1000 BERLIN 65, GERMANY
[2] AS FERROSAN, DK-2860 Soborg, DENMARK
关键词
D O I
10.1016/0361-9230(87)90099-2
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:309 / 318
页数:10
相关论文
共 35 条
  • [1] BETA-CARBOLINES AS LIGANDS OF THE BENZODIAZEPINE RECEPTOR
    MULLER, WE
    [J]. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1982, 363 (11): : 1284 - 1285
  • [2] BIDIRECTIONAL EFFECTS ON ANXIETY OF BETA-CARBOLINES ACTING AS BENZODIAZEPINE RECEPTOR LIGANDS
    STEPHENS, DN
    KEHR, W
    SCHNEIDER, HH
    BRAESTRUP, C
    [J]. NEUROPHARMACOLOGY, 1984, 23 (7B) : 879 - 880
  • [3] BETA-CARBOLINES - ENDOGENOUS LIGANDS FOR THE BENZODIAZEPINE RECEPTOR
    OGAWA, N
    MORI, A
    [J]. FOLIA PSYCHIATRICA ET NEUROLOGICA JAPONICA, 1984, 38 (03): : 207 - 211
  • [4] ARE THE PHARMACOLOGICAL ACTIONS OF BETA-CARBOLINES MEDIATED BY BENZODIAZEPINE RECEPTORS
    ROMMELSPACHER, H
    BRUNING, G
    [J]. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1981, 362 (10): : 1298 - 1299
  • [5] SYNTHESIS OF NOVEL 3-SUBSTITUTED BETA-CARBOLINES AS BENZODIAZEPINE RECEPTOR LIGANDS - PROBING THE BENZODIAZEPINE RECEPTOR PHARMACOPHORE
    ALLEN, MS
    HAGEN, TJ
    TRUDELL, ML
    CODDING, PW
    SKOLNICK, P
    COOK, JM
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) : 1854 - 1861
  • [6] BENZODIAZEPINE ANTAGONISM BY HARMANE AND OTHER BETA-CARBOLINES INVITRO AND INVIVO
    ROMMELSPACHER, H
    NANZ, C
    BORBE, HO
    FEHSKE, KJ
    MULLER, WE
    WOLLERT, U
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (03) : 409 - 416
  • [7] BETA-CARBOLINES - SYNTHESIS AND NEUROCHEMICAL AND PHARMACOLOGICAL ACTIONS ON BRAIN BENZODIAZEPINE RECEPTORS
    CAIN, M
    WEBER, RW
    GUZMAN, F
    COOK, JM
    BARKER, SA
    RICE, KC
    CRAWLEY, JN
    PAUL, SM
    SKOLNICK, P
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (09) : 1081 - 1091
  • [8] BETA-CARBOLINES - SYNTHESIS, NEUROCHEMICAL, AND PHARMACOLOGICAL ACTIONS ON BRAIN BENZODIAZEPINE RECEPTORS
    CAIN, M
    GUZMAN, F
    LARSCHEID, P
    COOK, JM
    SCHWERI, M
    PAUL, S
    MENDELSON, W
    SKOLNICK, P
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1982, 184 (SEP): : 76 - MEDI
  • [9] INTERACTIONS OF BENZODIAZEPINES AND BETA-CARBOLINES WITH A HISTIDINE RESIDUE OF THE BENZODIAZEPINE RECEPTOR
    LAMBOLEZ, B
    DESCHAMPS, CM
    ROSSIER, J
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1989, 15 (02) : 145 - 152
  • [10] BETA-CARBOLINES AS BENZODIAZEPINE RECEPTOR LIGANDS .1. SYNTHESIS AND BENZODIAZEPINE RECEPTOR INTERACTION OF ESTERS OF BETA-CARBOLINE-3-CARBOXYLIC ACID
    LIPPKE, KP
    SCHUNACK, WG
    WENNING, W
    MULLER, WE
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (04) : 499 - 503