THROMBIN ACTIVE-SITE INHIBITORS

被引:89
|
作者
DAS, J [1 ]
KIMBALL, SD [1 ]
机构
[1] BRISTOL MYERS SQUIBB CO, PHARMACEUT RES INST, PRINCETON, NJ 08543 USA
关键词
D O I
10.1016/0968-0896(95)00104-O
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
Development of small molecule thrombin active site inhibitors has been an area of intense research. A brief review on recent progress and challenges is outlined.
引用
收藏
页码:999 / 1007
页数:9
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