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SCH-28080 IS A LUMENALLY ACTING, K+-SITE INHIBITOR OF THE GASTRIC (H+ + K+)-ATPASE
被引:72
|
作者
:
KEELING, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
KEELING, DJ
[
1
]
LAING, SM
论文数:
0
引用数:
0
h-index:
0
机构:
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
LAING, SM
[
1
]
SENNBILFINGER, J
论文数:
0
引用数:
0
h-index:
0
机构:
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
SENNBILFINGER, J
[
1
]
机构
:
[1]
BYK GULDEN LOMBERG CHEM FABR GMBH,D-7750 KONSTANTZ,FED REP GER
来源
:
BIOCHEMICAL PHARMACOLOGY
|
1988年
/ 37卷
/ 11期
关键词
:
D O I
:
10.1016/0006-2952(88)90586-2
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
引用
收藏
页码:2231 / 2236
页数:6
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BINDING OF THE (H+ + K+)-ATPASE INHIBITOR, SCH-28080, TO GASTRIC MEMBRANE PREPARATIONS
KEELING, DJ
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SK&F RES LTD,WELWYN AL6 9AR,HERTS,ENGLAND
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KEELING, DJ
[J].
BIOCHEMICAL SOCIETY TRANSACTIONS,
1987,
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[2]
SCH-28080 IS A MORE SELECTIVE INHIBITOR THAN SCH-32651 AT THE K+ SITE OF GASTRIC K+/H+-ATPASE
BEIL, W
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SK-AND-F-96067 IS A REVERSIBLE, LUMENALLY ACTING INHIBITOR OF THE GASTRIC (H+ + K+)-ATPASE
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LEACH, CA
[J].
BIOCHEMICAL PHARMACOLOGY,
1991,
42
(01)
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[4]
INHIBITION OF H+K+ ATPASE BY SCH-28080 AND SCH-32651
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[J].
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112
(02)
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[5]
SCH 28080, A REVERSIBLE (H+ + K+)-ATPASE INHIBITOR, IS PREFERENTIALLY ACTIVE IN THE PROTONATED FORM
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[J].
BIOCHEMICAL SOCIETY TRANSACTIONS,
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[6]
Involvement of glutamic acid 820 in K+ and SCH 28080 binding to gastric H+,K+-ATPase
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[J].
NA/K-ATPASE AND RELATED TRANSPORT ATPASES: STRUCTURE, MECHANISM, AND REGULATION,
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PHOSPHORYLATION OF H+/K+-ATPASE BY INORGANIC-PHOSPHATE - THE ROLE OF K+ AND SCH 28080
VANDERHIJDEN, HTWM
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SCH-28080 IS A HIGHLY SELECTIVE COMPETITOR FOR THE PARIETAL-CELL PROTON PUMP K+-SITE
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The H+/K+ ATPase Inhibitor SCH-28080 Inhibits Insulin Secretion and Induces Cell Death in INS-1E Rat Insulinoma Cells
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[J].
CELLULAR PHYSIOLOGY AND BIOCHEMISTRY,
2017,
43
(03)
: 1037
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1051
[10]
INHIBITION OF GASTRIC H+,K+-ATPASE AND ACID-SECRETION BY SCH-28080, A SUBSTITUTED PYRIDYL(1,2A)IMIDAZOLE
WALLMARK, B
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0
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BRIVING, C
论文数:
0
引用数:
0
h-index:
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机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
BRIVING, C
FRYKLUND, J
论文数:
0
引用数:
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h-index:
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机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
FRYKLUND, J
MUNSON, K
论文数:
0
引用数:
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h-index:
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机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
MUNSON, K
JACKSON, R
论文数:
0
引用数:
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h-index:
0
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VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
JACKSON, R
MENDLEIN, J
论文数:
0
引用数:
0
h-index:
0
机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
MENDLEIN, J
RABON, E
论文数:
0
引用数:
0
h-index:
0
机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
RABON, E
SACHS, G
论文数:
0
引用数:
0
h-index:
0
机构:
VET ADM WADSWORTH HOSP,CTR ULCER RES & EDUC,LOS ANGELES,CA 90073
SACHS, G
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1987,
262
(05)
: 2077
-
2084
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