RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE

被引:203
|
作者
BOGER, J
PAYNE, LS
PERLOW, DS
LOHR, NS
POE, M
BLAINE, EH
ULM, EH
SCHORN, TW
LAMONT, BI
LIN, TY
KAWAI, M
RICH, DH
VEBER, DF
机构
[1] MERCK SHARP & DOHME RES LABS, RAHWAY, NJ 07065 USA
[2] UNIV WISCONSIN, SCH PHARM, MADISON, WI 53706 USA
关键词
D O I
10.1021/jm00150a007
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
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页码:1779 / 1790
页数:12
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