A simple and efficient synthesis of 2-aryl-substituted benzimidazoles

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作者
Xiangming Han
Huiqiang Ma
Yulu Wang
机构
[1] Henan Normal University,College of Chemistry and Environmental Science
[2] Pingyuan University,Department of Chemistry and Environmental Engineering
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关键词
Benzimidazole; Azole; Aromatic Aldehyde; Sulfamic Acid; Easy Purification;
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摘要
Sodium hydrogen sulfite was used to promote condensation of o-phenylenediamine with aromatic aldehydes in dimethylformamide to obtain the corresponding 2-arylbenzimidazoles. The procedure is simple and convenient, and it implies inexpensive promoter and is characterized by short reaction time and easy purification of the final products.
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