Tetrazoles: LIII. Microwave-activated acylation of 5-substituted tetrazoles

被引：0
|
作者：
Yu. A. Efimova
T. V. Artamonova
G. I. Koldobskii
机构：
[1] St. Petersburg State Institute of Technology,
来源：
Russian Journal of Organic Chemistry | 2008年 / 44卷
关键词：
Microwave Irradiation; Acetic Anhydride; Oxadiazole; Aqueous Sodium Hydroxide; Microwave Activation;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
The acylation of 5-aryl(hetaryl)tetrazoles with acetic and benzoic anhydrides under microwave irradiation gave the corresponding 2-substituted 5-methyl-and 5-phenyl-1,3,4-oxadiazoles in high yields. The use of microwave activation reduces the reaction temperature by 30–40°C and shortens the reaction time by a factor of 5 to 7.
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