In silico discovery and validation of potent small-molecule inhibitors targeting the activation function 2 site of human oestrogen receptor α

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作者
Kriti Singh
Ravi Shashi Nayana Munuganti
Eric Leblanc
Yu Lun Lin
Euphemia Leung
Nada Lallous
Miriam Butler
Artem Cherkasov
Paul S Rennie
机构
[1] University of British Columbia,Vancouver Prostate Centre
[2] University of Auckland,Auckland Cancer Society Research Centre
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MCF7 Cell; Root Mean Square Deviation; Virtual Screening; Fulvestrant; Carbohydrazide;
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