Benzazoles 5*. Synthesis and arylsulfonylation of 1-hydroxymethylbenzimidazole

被引：0
|
作者：
K. B. Abdireimov
N. S. Mukhamedov
M. Zh. Aiymbetov
Kh. M. Shakhidoyatov
机构：
[1] S. Yu. Yunusov Institute of the Chemistry of Plant Substances,
[2] Academy of Sciences of Uzbekistan,undefined
来源：
Chemistry of Heterocyclic Compounds | 2012年 / 48卷
关键词：
1-arylsulfonylbenzimidazoles; 1-hydroxymethylbenzimidazole; arylsulfonylation; hydroxy-methylation; deformylation;
D O I：
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中图分类号：
学科分类号：
摘要：
1-Hydroxymethylbenzimidazole was synthesized by the reaction of benzimidazole with formaldehyde. Arylsulfonylation of the former in the presence of triethylamine occurred anomalously with deformylation to give 1-arylsulfonylbenzimidazoles in place of the expected 1-arylsulfonyloxymethyl-benzimidazoles.
引用
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页码：458 / 461
页数：3
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