Mass Balance, Metabolism, and Excretion of Cenobamate, a New Antiepileptic Drug, After a Single Oral Administration in Healthy Male Subjects

被引:0
|
作者
Laurent Vernillet
Stephen A. Greene
Hong Wook Kim
Susan M. Melnick
Kelli Glenn
机构
[1] SK Life Science,Department of Clinical Pharmacology
[2] Inc,Department of Toxicology
[3] SK Life Science,undefined
[4] Inc,undefined
关键词
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:513 / 522
页数:9
相关论文
共 50 条
  • [1] Mass Balance, Metabolism, and Excretion of Cenobamate, a New Antiepileptic Drug, After a Single Oral Administration in Healthy Male Subjects
    Vernillet, Laurent
    Greene, Stephen A.
    Kim, Hong Wook
    Melnick, Susan M.
    Glenn, Kelli
    EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2020, 45 (04) : 513 - 522
  • [2] ABSORPTION, DISTRIBUTION, METABOLISM, AND EXCRETION OF THE NOVEL ANTIEPILEPTIC DRUG CENOBAMATE: MASS BALANCE FOLLOWING ORAL ADMINISTRATION IN HEALTHY MALE SUBJECTS
    Glenn, Kelli J.
    Greene, Stephen
    Kim, Hong-Wook
    Melnick, Susan M.
    Vernillet, Laurent
    DRUG METABOLISM AND PHARMACOKINETICS, 2020, 35 (01) : S69 - S69
  • [3] MASS BALANCE AND METABOLITE IDENTIFICATION OF VALEMETOSTAT AFTER A SINGLE ORAL ADMINISTRATION IN HEALTHY MALE SUBJECTS
    Inaba, S.
    Kazui, M.
    Shimizu, T.
    Craveiro, T.
    Abutarif, M.
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 2023, 113 : S57 - S57
  • [4] THE MASS BALANCE RECOVERY, ABSORPTION, METABOLISM, AND EXCRETION OF [14C]-ORVEPITANT IN HEALTHY MALE SUBJECTS AFTER ORAL DOSING: CLINICAL CONDUCT & MASS BALANCE
    Shaw, Iain
    Singh, Nand
    Melbourne, Sue
    Cooke, Ray
    Lock, Ruth
    Pawsey, Steve
    DRUG METABOLISM AND PHARMACOKINETICS, 2024, 55
  • [5] The Mass Balance Recovery, Absorption, Metabolism, and Excretion of [14C]Orvepitant in Healthy Male Subjects After Oral Dosing: Radiosynthesis
    Carver, D.
    Cousin, P.
    Martos, J.
    Craig, J.
    Lawrence, R.
    Shaw, I.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2024, 67 (10): : 354 - 354
  • [6] THE MASS BALANCE, RECOVERY, ABSORPTION, METABOLISM, AND EXCRETION OF [14C]-ORVEPITANT IN HEALTHY MALE SUBJECTS AFTER ORAL DOSING: METABOLITE CHARACTERISATION
    Colato, Dimitri
    Bordini, Ellenia
    Cufari, Domenico
    Lock, Ruth
    Pawsey, Steve
    Melbourne, Sue
    Shaw, Iain
    DRUG METABOLISM AND PHARMACOKINETICS, 2024, 55
  • [7] Absorption, Metabolism, and Excretion of [14C]-Labeled Anaprazole: A New Proton Pump Inhibitor, After a Single Oral Administration in Healthy Chinese Male Subjects
    Xie, Lijun
    Xu, Yanjun
    Liu, Wei
    Zhou, Chen
    Guo, Lian
    Zhou, Sufeng
    Zhang, Chen
    Chen, Juan
    Zhu, Bei
    Ding, Sijia
    Li, Huan
    Zhang, Lingling
    Wang, Li
    Xu, Lingmei
    Shao, Feng
    Wang, Lu
    CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2024, 13 (10): : 1115 - 1122
  • [8] Pharmacokinetics, metabolism and excretion of 14C-ragaglitazar after a single oral dose to healthy male subjects
    Vanggaard, J
    Wassmann, O
    Andersen, MP
    Skrumsager, BK
    DIABETES, 2002, 51 : A490 - A490
  • [9] 14C-ragaglitazar:: pharmacokinetics, metabolism and excretion after a single oral dose to healthy male subjects
    Vanggaard, J
    Wassmann, O
    Andersen, MP
    Skrumsager, BK
    DIABETOLOGIA, 2002, 45 : A232 - A232
  • [10] Mass Balance and Absorption, Distribution, Metabolism, and Excretion Properties of Balcinrenone following Oral Administration in Combination with Intravenous Microtracer in Healthy Subjects
    Lindmark, Bo
    Li, Xue-Qing
    Bhattacharya, Chandrali
    Housler, Greggory
    Heijer, Maria
    Bragg, Ryan A.
    Granfors, Malin
    Pelay-Gimeno, Marta
    Vaes, Wouter H. J.
    Menakuru, Somasekhara
    Pizzato, Patricia Ely
    Ericsson, Hans
    Johansson, Susanne
    DRUG METABOLISM AND DISPOSITION, 2023, 51 (08) : 995 - 1004