The total large-scale synthesis of argiopine

被引:0
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作者
A. A. Formanovsky
I. S. Popova
I. V. Mikhura
机构
[1] Russian Academy of Sciences,Shemyakin
关键词
argiopine; polymethylenepolyamines; synthesis;
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学科分类号
摘要
The total large-scale synthesis of a natural toxin argiopine, a polymethylenepolyamine derivative, was developed. It consisted of 26 stages and included three key block schemes. Most of the stages proceeded quantitatively, which excluded the necessity of using the chromatographic separation of intermediates.
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页码:752 / 758
页数:6
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