Nucleophilic substitution in 1,5-benzodiazepin-2-ones

被引：0
|
作者：
Bozhanov V.I. [1 ]
Ivonin S.P. [1 ]
机构：
[1] Dnepropetrovsk State University, UKR
来源：
Chemistry of Heterocyclic Compounds | 2000年 / 36卷 / 12期
关键词：
1,5-benzodiazepin-2-ones; Bromination; phase-transfer catalysis; Nucleophilic substitution; Thiazolo[4,5-b][1,5]benzodiazepine;
D O I：
10.1023/A:1017578614850
中图分类号：
学科分类号：
摘要：
The reaction of 3-bromo-4-phenyl-2,3-dihydro-1H -1,5-benzodiazepin-2-one with cyclic amines gives 3-aminoalkyl-4-phenyl-2,3-dihydro-1H-1,5-benzodiazepin-2-one. Thiazolo[4, 5-b][1,5]benzodiazepine was isolated along with the substitution product when thiourea was used.
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收藏
页码：1446 / 1448
页数：2
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