Positive-allosteric modulation of the 5-HT2C receptor: implications for neuropsychopharmacology and neurotherapeutics

被引:0
|
作者
Jia Zhou
Kathryn A. Cunningham
机构
[1] University of Texas Medical Branch,Center for Addiction Research and Department of Pharmacology and Toxicology
来源
Neuropsychopharmacology | 2019年 / 44卷
关键词
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:230 / 231
页数:1
相关论文
共 50 条
  • [1] Positive-allosteric modulation of the 5-HT2C receptor: implications for neuropsychopharmacology and neurotherapeutics
    Zhou, Jia
    Cunningham, Kathryn A.
    NEUROPSYCHOPHARMACOLOGY, 2019, 44 (01) : 230 - 231
  • [2] Serotonin (5-HT) 5-HT2C receptor (5-HT2CR) positive allosteric modulators as novel neurotherapeutics
    Wild, Christopher
    McAllister, Carrie E.
    Wold, Eric A.
    Ding, Chunyong
    Anastasio, Noelle C.
    Fox, Robert G.
    Stutz, Sonja J.
    Chen, Haiying
    Tomlinson, Suzanne
    Cunningham, Kathryn
    Zhou, Jia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251
  • [3] Positive allosteric modulator of the human 5-HT2C receptor
    Bin Im, W
    Chio, CL
    Alberts, GL
    Dinh, DM
    MOLECULAR PHARMACOLOGY, 2003, 64 (01) : 78 - 84
  • [4] A Positive Allosteric Modulator of the Serotonin 5-HT2c Receptor for Obesity
    Garcia-Carceles, Javier
    Decara, Juan M.
    Vazquez-Villa, Henar
    Rodriguez, Ramon
    Codesido, Eva
    Cruces, Jacobo
    Brea, Jose
    Loza, Maria I.
    Alen, Francisco
    Botta, Joaquin
    McCormick, Peter J.
    Ballesteros, Juan A.
    Benhamu, Bellinda
    Rodriguez de Fonseca, Fernando
    Lopez-Rodriguez, Maria L.
    JOURNAL OF MEDICINAL CHEMISTRY, 2017, 60 (23) : 9575 - 9584
  • [5] Discovery of Novel Oleamide Analogues as Brain-Penetrant Positive Allosteric Serotonin 5-HT2C Receptor and Dual 5-HT2C/5-HT2A Receptor Modulators
    Chen, Jianping
    Garcia, Erik J.
    Merritt, Christina R.
    Zamora, Joshua C.
    Bolinger, Andrew A.
    Pazdrak, Konrad
    Stafford, Susan J.
    Mifflin, Randy C.
    Wold, Eric A.
    Wild, Christopher T.
    Chen, Haiying
    Anastasio, Noelle C.
    Cunningham, Kathryn A.
    Zhou, Jia
    JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (14) : 9992 - 10009
  • [6] Discovery of novel potent and selective agonists of the serotonin (5-HT) 5-HT2C receptor as neurotherapeutics
    Mack, Helmut
    Backfisch, Gisela
    Blaich, Guenter
    Braje, Wilfried
    Erhard, Thomas
    Haupt, Andreas
    Kling, Andreas
    Lakics, Viktor
    Lynch, James
    Mugnaini, Manolo
    Pohlki, Frauke
    Relo, Ana
    Schaefer, Kai
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253
  • [7] 5-HT2C receptor modulation and the treatment of obesity
    Bickerdike, MJ
    Vickers, SP
    Dourish, CT
    DIABETES OBESITY & METABOLISM, 1999, 1 (04): : 207 - 214
  • [8] Design, synthesis, and pharmacological evaluation of novel positive allosteric modulators (PAMs) of 5-HT2C receptor
    Ding, Chunyong
    Zhang, Gongliang
    Anastasio, Noelle C.
    Moncrief', Scott
    Carbonaro, Theresa M.
    Fox, Robert G.
    Stutz, Sonja
    Wild, Christopher
    Smith, Thressa D.
    Hartley, Rachel M.
    White, Mark A.
    Cunningham, Kathryn A.
    Zhou, Jia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247
  • [9] Pharmacological Evaluations of a Novel Chemical Series of Serotonin 5-HT2C Receptor (5-HT2CR) Positive Allosteric Modulators
    Anastasio, Noelle
    Wold, Eric
    Garcia, Erik
    Pazdrak, Konrad
    Chen, Jianping
    Wild, Christopher
    Zhou, Jia
    Cunningham, Kathryn
    NEUROPSYCHOPHARMACOLOGY, 2019, 44 (SUPPL 1) : 200 - 201
  • [10] Discovery of 4-undecylpiperidine-2-carboxamides as selective positive allosteric modulators of the serotonin (5-HT) 5-HT2C receptor
    Wold, Eric
    Wild, Christopher
    McAllister, Carrie
    Crawford, Claudia
    Ding, Ye
    Anastasio, Noelle
    Fox, Robert
    Stutz, Sonja
    Hartley, Rachel
    Chen, Haiying
    White, Mark
    Cunningham, Kathryn
    Zhou, Jia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252