Synthesis of N-substituted derivatives of (5-amino-2-methyl-1H-indol-3-YL)acetic acid

被引：0
|
作者：
Maklakov S.A. [1 ]
Smushkevich Yu.I. [2 ]
Magedov I.V. [3 ]
机构：
[1] Novomoskovsk Institute, D. I. Mendeleev Russian University of Chemical Technology
[2] D. I. Mendeleev Russian University of Chemical Technology
[3] Moscow K. A. Timiryazev Agricultural Academy
来源：
Chemistry of Heterocyclic Compounds | 2002年 / 38卷 / 5期
关键词：
(5-amino-2-methyl-1H-indol-3-yl)acetic acid; Fischer reaction; Indole; Indomethacin; N-(4-hydrazinophenyl)acetamide;
D O I：
10.1023/A:1019500911047
中图分类号：
学科分类号：
摘要：
A method has been developed for obtaining indole compounds containing an amino group in the benzene ring by the indolization of ethyl levulinate p-acetaminophenylhydrazone. A series of derivatives of (5-amino-2-methyl-1H-indol-3-yl)acetic acid at the 5-amino group has been synthesized.
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页码：539 / 542
页数：3
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