Synthesis of Some New Heterocyclic Compounds Derived from 3-Formylchromones and Their Antimicrobial Evaluation

被引：0

作者：

A. Bari

S. S. Ali

A. Kadi

I. A. Hashmi

S. W. Ng

机构：

[1] King Saud University,Department of Pharmaceutical Chemistry, College of Pharmacy

[2] King Saud University,Research Center, College of Pharmacy

[3] University of Karachi,Department of Chemistry

[4] University of Malaya,Department of Chemistry

来源：

Chemistry of Heterocyclic Compounds | 2014年 / 49卷

关键词：

3-formylchromone; pyranopyrones; antimicrobial activity; enzyme inhibitors; Knoevenagel–Cope reaction; pharmacophore; urease inhibitory;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

The synthesis and antimicrobial evaluation of a series of chromone-linked substituted heterocyclic derivatives is described. The condensation of 3-formylchromone with acetoacetamide under Knoevenagel–Cope reaction conditions was also explored, and the condensation with 4-hydroxy-6-methyl-2H-pyran-2-one constitutes a facile route to pyranopyrone fused systems. Most of the compounds exhibit good antimicrobial properties.

引用

页码：1723 / 1731

页数：8

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