PARA-AMINOSALICYLIC ACID (PAS) CHARACTERIZED AS A SUBSTRATE OF OCT1 AND OCT2 AND OAT1 AND OAT3 TRANSPORTER AND OCT1/2 POLYMORPHISM EFFECT, IN VITRO

被引:0
|
作者
Parvez, M. D. Masud [1 ,2 ]
Jung, Jin-Ah [3 ]
Shin, Ho Jung [1 ,2 ]
Kaisar, Nazia [1 ,2 ]
Hasanuzzaman, M. D. [1 ,2 ]
Kim, Dong-Hyun [1 ,2 ]
Shin, Jae-Gook [1 ,2 ,3 ]
机构
[1] Inje Univ, Coll Med, Dept Pharmacol, Busan, South Korea
[2] Inje Univ, Coll Med, Pharmacogen Res Ctr, Busan, South Korea
[3] Inje Univ, Busan Paik Hosp, Dept Clin Pharmacol, Busan, South Korea
关键词
D O I
10.1016/j.dmpk.2016.10.389
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
P263
引用
收藏
页码:S102 / S102
页数:1
相关论文
共 50 条
  • [1] PARA-AMINOSALYCYLIC ACID (PAS) CHARACTERIZED AS A SUBSTRATE OF OCT1 AND OCT2 AND OAT1 AND OAT3 TRANSPORTER, IN VITRO.
    Masud, P. Md.
    Jung, J.
    Choi, H.
    Shin, H.
    Kim, D.
    Shin, J.
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 2016, 99 : S97 - S97
  • [2] In vitro interaction of clopidogrel and its hydrolysate with OCT1, OCT2 and OAT1
    Li, Liping
    Song, Feifeng
    Tu, Meijuan
    Wang, Kai
    Zhao, Lei
    Wu, Xiaodan
    Zhou, Hui
    Xia, Zongling
    Jiang, Huidi
    INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2014, 465 (1-2) : 5 - 10
  • [3] Molecular Properties of Drugs Interacting with SLC22 Transporters OAT1, OAT3, OCT1, and OCT2: A Machine-Learning Approachs
    Liu, Henry C.
    Goldenberg, Anne
    Chen, Yuchen
    Lun, Christina
    Wu, Wei
    Bush, Kevin T.
    Balac, Natasha
    Rodriguez, Paul
    Abagyan, Ruben
    Nigam, Sanjay K.
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2016, 359 (01): : 215 - 229
  • [4] Inhibition of human OCT1, OCT2, MATE1, OAT1 and NTCP mediated uptake by pesticides
    Kuehne, A.
    Floerl, S.
    Halpape, R.
    Hagos, Y.
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2018, 391 : S72 - S73
  • [5] Differential substrate specificity of rabbit OCT1 and OCT2
    Kaewmokul, S
    Chatsudthipong, V
    Wright, SH
    FASEB JOURNAL, 2002, 16 (04): : A459 - A459
  • [6] The interaction of steviol with rabbit OCT1 and OCT2
    Chatsudthipong, V
    Lungkaphin, A
    Kaewmokul, S
    FASEB JOURNAL, 2003, 17 (04): : A476 - A476
  • [7] Renal uptake of substrates for organic anion transporters Oat1 and Oat3 and organic cation transporters Oct1 and Oct2 is altered in rats with adenine-induced chronic renal failure
    Komazawa, Hiroki
    Yamaguchi, Hiroaki
    Hidaka, Kazuhiro
    Ogura, Jiro
    Kobayashi, Masaki
    Iseki, Ken
    JOURNAL OF PHARMACEUTICAL SCIENCES, 2013, 102 (03) : 1086 - 1094
  • [8] Substrates and Inhibitors of the Organic Cation Transporter 3 and Comparison with OCT1 and OCT2
    Gebauer, Lukas
    Jensen, Ole
    Brockmoeller, Juergen
    Duecker, Christof
    JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (18) : 12403 - 12416
  • [9] Effect of OCT1 and OCT1 polymorphism on the hepatocellular uptake and the pharmacokinetics of proguanil
    Seitz, T.
    Matthaei, J.
    Tann, A.
    Brockmoeller, J.
    Tzvetkov, M.
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2017, 390 : S75 - S75
  • [10] Organic cation transporters (OCT1, OCT2 and OCT3) and organic anion transporter (OAT3) mediate the uptake of duodenal ulcerogen cysteamine in intestinal epithelial cells (IEC-6)
    Khomenko, Tetyana
    Tolstanova, Ganna
    Chen, Longchuan
    Deng, Xiaoming
    Said, Hamid M.
    Szabo, Sander
    GASTROENTEROLOGY, 2007, 132 (04) : A575 - A576