Design and synthesis of lysine-targeted covalent inhibitors of HSP72

被引：0
|
作者：
Pettinger, Jonathan [1 ]
Le Bihan, Yann-Vai [1 ]
Powers, Marissa [1 ]
Widya, Marcella [2 ]
van Montfort, Rob [1 ]
Jones, Keith [1 ]
Cheeseman, Matthew [1 ]
机构：
[1] Inst Canc Res, Div Canc Therapeut, London, England
[2] Novartis Inst BioMed Res, Berkeley, CA USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2018年 / 255卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
16
引用
收藏
页数：2
相关论文
共 50 条
  • [1] Design and synthesis of lysine-56 targeting covalent inhibitors of HSP72
    Pettinger, Jonathan
    Cheeseman, Matthew
    Le Bihan, Yann-Vai
    Widya, Marcella
    van Montfort, Rob
    Jones, Keith
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253
  • [2] Kinetic Optimization of Lysine-Targeting Covalent Inhibitors of HSP72
    Pettinger, Jonathan
    Carter, Michael
    Jones, Keith
    Cheeseman, Matthew D.
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (24) : 11383 - 11398
  • [3] Lysine-targeted covalent inhibitors and chemoproteomic probes
    Taunton, Jack
    [J]. MOLECULAR & CELLULAR PROTEOMICS, 2019, 18 (08) : S20 - S20
  • [4] Strategic design of lysine-targeted irreversible covalent NDM-1 inhibitors
    Ma, Youzhen
    Liang, Yongxi
    Guo, Menglu
    Min, Delin
    Zheng, Lulu
    Tang, Yun
    Sun, Xun
    [J]. CHINESE CHEMICAL LETTERS, 2023, 34 (07)
  • [5] Strategic design of lysine-targeted irreversible covalent NDM-1 inhibitors
    Youzhen Ma
    Yongxi Liang
    Menglu Guo
    Delin Min
    Lulu Zheng
    Yun Tang
    Xun Sun
    [J]. Chinese Chemical Letters, 2023, 34 (07) : 172 - 176
  • [6] Lysine-Targeted Inhibitors and Chemoproteomic Probes
    Cuesta, Adolfo
    Taunton, Jack
    [J]. ANNUAL REVIEW OF BIOCHEMISTRY, VOL 88, 2019, 88 : 365 - 381
  • [7] Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking
    Wan, Xiaobo
    Yang, Tangpo
    Cuesta, Adolfo
    Pang, Xiaming
    Balius, Trent E.
    Irwin, John J.
    Shoichet, Brian K.
    Taunton, Jack
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2020, 142 (11) : 4960 - 4964
  • [8] Tuning residence time with lysine-targeted, reversible covalent probes
    Yang, Tangpo
    Cuesta, Adolfo
    Wan, Xiaobo
    Taunton, Jack
    [J]. MOLECULAR & CELLULAR PROTEOMICS, 2019, 18 (08) : S52 - S52
  • [9] Identification of novel allosteric HSP72 inhibitors
    Traynor, Hannah
    Burke, Rosemary
    Le Bihan, Yann-Vai
    Collins, Ian
    Van Montfort, Rob
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253
  • [10] Lysine-Targeted Reversible Covalent Ligand Discovery for Proteins via Phage Display
    Zheng, Mengmeng
    Chen, Fa-Jie
    Li, Kaicheng
    Reja, Rahi M.
    Haeffner, Fredrik
    Gao, Jianmin
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 144 (34) : 15885 - 15893
12345